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{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-3-ylmethyl)amine
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propyl acetate
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
3-{[6-(propan-2-yl)pyrimidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[2-(4-{[3-(1,3-benzothiazol-2-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclopropanecarbonylpiperidin-3-yl)piperazine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)pyridin-2-amine
4-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]thiophene-2-carboxamide
3-(4-fluorophenyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
8-(2-fluorobenzoyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(3R,4S)-1-{[4-(2-methylpropyl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]urea
2-amino-6-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
4-(piperidin-4-yl)-6-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidine
1-(3,5-difluorophenyl)-N-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3S,4R)-1-(2-methanesulfonylethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-[1-(3-methylbutyl)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
1-[2-(ethylsulfanyl)phenyl]-3-(oxolan-2-ylmethyl)-3-(thiophen-3-ylmethyl)urea
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-1,3-thiazole-5-carboxamide
3,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzofuran-2-carboxamide
N-(2-methoxyethyl)-4-methyl-3-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
methyl (1R,3S,3aR,6aS)-1-benzyl-5-methyl-3-(1-methyl-1H-imidazol-5-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-(2-phenylethyl)-3-(propan-2-yl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-[(1R,3S,3aS,6aR)-3-(1-ethyl-1H-imidazol-5-yl)-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
N-ethyl-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-fluorophenyl)-3-phenylpropanamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]piperidine
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
[2-(4-methoxyphenyl)ethyl][(1-methyl-1H-indol-3-yl)methyl][(1-methylpiperidin-4-yl)methyl]amine
7-(2-amino-6-methoxypyrimidin-4-yl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-[(dimethylamino)methyl]furan-2-carboxamide
(1S,4S)-2-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-azabicyclo[2.2.1]heptane
2-(4-fluorophenyl)-N-(2-oxopiperidin-3-yl)imidazo[1,2-a]pyridine-6-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]benzamide
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-methyl-1,3-oxazole-5-carboxamide
2-{2-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-{5-cyclopropyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2,5-dimethylthiophen-3-yl)pyrimidine
5-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-methanesulfonamido-N-[(3R,4S)-4-propyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]acetamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1,2,3,6-tetrahydropyridin-4-yl}propan-2-yl)acetamide
3-[2-(3-methoxyphenyl)ethyl]-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine
4-(1H-imidazol-1-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylic acid
(3E)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}pent-3-enamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]benzamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(1,2,5-thiadiazole-3-carbonyl)-1,4-diazepan-2-one