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2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-(3-ethylpiperazin-1-yl)ethan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylpiperidine-3-carboxamide
4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyrimidin-2-amine
N-(2-hydroxyethyl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-(thiophen-2-ylmethyl)benzamide
(1S,5R)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
N-(3-methylbutyl)-2-oxo-1-phenylpyrrolidine-3-carboxamide
1-[2-(2-chlorophenoxy)ethyl]-3-(methoxymethyl)pyrrolidine
(4aS,8aR)-6-(4,6-dimethoxypyrimidin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
9-methoxy-7-(6-methoxypyridazin-3-yl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
3-(2,8-dimethylquinoline-3-carbonyl)-3,9-diazaspiro[5.5]undecane
(2S,4R)-4-[2-(5-acetylthiophen-3-yl)acetamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(2-ethyl-1H-imidazol-1-yl)propanamide
1-(4-methoxyphenyl)-4-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
6-[2-(benzyloxy)ethyl]-2-methyl-[1,2,4]triazolo[1,5-a]pyridine
2-{4-[1-(pyrimidin-2-yl)piperidin-4-yl]piperazin-1-yl}pyrazine
N-[2-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)ethyl]acetamide
9-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-6-oxa-9-azaspiro[4.5]decane
1-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopropane-1-carbonitrile
7-(cyclopropylmethyl)-2-(quinolin-8-ylmethyl)-2,7-diazaspiro[4.5]decane
2-(2-ethoxyphenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
1-(cyclohexylmethyl)-5-(1,4-dioxan-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
methyl 1-[(3S,5S)-1-(cyclohexylmethyl)-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(2-phenylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
methyl 4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}benzoate
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
(2S)-2-amino-N-(1-benzothiophen-5-ylmethyl)-3-(4-hydroxyphenyl)propanamide
2-phenyl-N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
6-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
6-methyl-2-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
[(8-methoxyquinolin-2-yl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-ethyl-N-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]pyrrolidin-3-yl}acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
3-(4-hydroxyphenyl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]morpholine-2-carboxamide
2,2-dimethyl-4-oxo-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-pyran-6-carboxamide
N-[(4-methylphenyl)methyl]-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrrolidin-2-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
3-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-diazinane-2,4-dione
2-[1-(cyclohexylmethyl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-(3,4-difluorophenyl)-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(cyclohex-3-en-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(2-methoxyphenyl)acetamide
1-(2-methoxyethyl)-2-(5-propylfuran-2-yl)-1H-imidazole
N-[(2-methoxyphenyl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine