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3-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidine-1-carbonyl]-6-methylpyridin-2-ol
N-(furan-2-ylmethyl)-N-methyl-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
4-methoxy-N-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzene-1-sulfonamide
1-methyl-N-(2-phenylethyl)-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-4-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}pyrimidin-2-amine
8-[2-(1H-1,2,4-triazol-5-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[(3R,4S)-1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
5-(3-methylbutyl)-5-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
2-ethyl-9-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
1-(3,5-dimethylphenyl)-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]piperazin-2-one
(4aS,7aR)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(1,2-oxazinan-2-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]pyridin-2-amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methanol
4-(4-fluoro-2-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
(2R,6S)-4-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-2,6-dimethylmorpholine
1-(2-methoxyethyl)-5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
4-[(6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridin-3-yl)methyl]morpholine
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]propanamide
7-(cyclopropylmethyl)-N-[(3-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(4aS,8aR)-N-ethyl-1-[2-(5-methylfuran-2-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
5-[2-(3-chlorophenoxy)propanoyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(oxolane-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N,N-diethyl-2-({2-oxo-4-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
2-(5-{5H,6H,7H-cyclopenta[b]pyridin-3-yl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl)acetic acid
5-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2,4-dimethylpyridine
4-(2-amino-1,3-thiazol-5-yl)-3-methyl-1-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
N-({4-hydroxy-1-[2-(1H-imidazol-1-yl)acetyl]azepan-4-yl}methyl)-2,5-dimethylfuran-3-carboxamide
3-({1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}carbamoyl)benzoic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3-ethoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,7S)-5-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(2-methanesulfonamidoethyl)-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-{2-[(3-fluorophenyl)methoxy]phenyl}-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
(3R,5S)-N3-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
methyl 3-acetamido-5-{[1-(3-methoxyphenyl)propan-2-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)propanamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
2-(carbamoylamino)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
4-(4-fluorophenyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,2,3,6-tetrahydropyridine
6-(2-methyl-1,3-thiazol-4-yl)-2-{3-[(4-methyl-3-oxopiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}acetamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
ethyl 4-{1-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxypyridine-3-carboxamide