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N-[2-(1H-indol-1-yl)ethyl]-N,2-dimethylpyrimidine-5-carboxamide
1-(prop-2-en-1-yl)-5-{[1-(pyrazin-2-yl)piperidin-4-yl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3aR,6aS)-N-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
7-(oxan-4-yl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
4-[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)sulfamoyl]-N-methylthiophene-2-carboxamide
1-cyclohexyl-5-(furan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-oxo-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-3,4-dihydrophthalazine-1-carboxamide
(4aS,7aR)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[benzyl(2-phenylethyl)amino]methyl}pyrrolidin-3-ol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclopropyl-1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-2-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
2-ethyl-3-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-[2-(1H-indol-3-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(2-ethylpyrimidine-5-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(3-fluorophenoxy)piperidine
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2,2-dimethyloxane-4-carboxamide
1-(3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)propan-1-one
3-(methoxymethyl)-N-[3-(piperidin-1-ylmethyl)phenyl]pyrrolidine-1-carboxamide
N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(1-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]acetamide
2-(2-methylpropyl)-8-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
methyl 4-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-1H-pyrazole-3-carboxylate
2-cyclopropanecarbonyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-methylpyrrolidine-3-carboxamide
2-{1-[(1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
(1R,3S)-7-[4-(3-fluorophenyl)benzoyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-(4-fluorophenyl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
{3-[(3-chlorophenyl)methyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl}methanol
9-(2-ethylpyridine-4-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[(3-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3,5-dimethylphenyl)-N-[(1R)-2-hydroxy-1-phenylethyl]propanamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamide
1-{[6-(2H-1,3-benzodioxol-5-yl)pyridin-3-yl]methyl}-4-methylpiperazine
phenyl (7S,9aR)-7-[(1R)-1-(benzyloxy)ethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-(cyclopropylmethyl)-3-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-3-hydroxypiperidin-2-one
3-(2-chlorophenyl)-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-methoxy-1-[3-(4-phenylbenzoyl)piperidin-1-yl]ethan-1-one
4-(2,2-dimethylpropyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
1-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-5-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]-1H-pyrrole-3-carbonitrile
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
1-(5-methyl-2,1,3-benzothiadiazol-4-yl)-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
5-({[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}methyl)-N-methylfuran-2-carboxamide