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dimethyl({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
1-(2-methylfuran-3-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-(cyclohexylmethyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(furan-2-carbonyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
2-(dimethyl-1,2-oxazol-4-yl)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
4-{[(3S,5R)-3-[(4-methylpiperazin-1-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}phenol
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[(1R)-1-phenylethyl]urea
(3aS,6aR)-N-(2-methylphenyl)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-(1-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-(2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine
2-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
N-(pyridin-4-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-methoxypyridazine
3-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
methyl 1-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidine-4-carboxylate
N-[(3,4-dimethoxyphenyl)methyl]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]-N-(pyridin-2-ylmethyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
1-benzyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
3-[(cyclopentylamino)methyl]-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methoxyphenol
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
(2,1,3-benzoxadiazol-5-ylmethyl)(benzylsulfamoyl)methylamine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
N-(pyridin-3-yl)quinoxaline-6-carboxamide
5-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoxaline
{3-[(4-fluorophenyl)methyl]-1-(4-methoxypyrimidin-2-yl)piperidin-3-yl}methanol
N-[3-(oxolan-3-yl)propyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
3-[(6-ethyl-4-methylquinolin-2-yl)amino]propane-1,2-diol
3-{1-[3-(3-chlorophenyl)propanoyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
6-(methoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrimidin-4-amine
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-(3-methoxyphenyl)-6-methyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrazine-2-carboxamide
7-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decane
2-cycloheptyl-4-{4-[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(1-acetylpiperidin-4-yl)-N-(1-benzylpyrrolidin-3-yl)propanamide
2-(3-cyclopropyl-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl)pyridine
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
5-[1-(2,2-diphenylethyl)piperidin-4-yl]-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
6-(2-chlorophenyl)-2-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-fluoro-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-5-sulfamoylbenzamide
1-[2-methoxy-4-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-[2-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
3-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)-N-phenylpropanamide