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(2S)-2-amino-1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-3-(1,3-thiazol-4-yl)propan-1-one
1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
N-(2-hydroxyethyl)-1-methyl-N-[(3-methylthiophen-2-yl)methyl]azepane-2-carboxamide
4-(1-{6-[(2S,5R)-2,5-dimethylpiperazin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)morpholine
6-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]naphthalen-2-ol
4-(4-{[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
2-[(methylsulfanyl)methyl]-4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
4-hydroxy-4-(1H-imidazol-1-ylmethyl)-N-[2-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
1-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-propylurea
8-cyclopropanecarbonyl-2-[3-(1H-pyrrol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(2-methoxypyridin-3-yl)-1H-pyrazole-3-carbonitrile
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(2,3-dimethoxyphenyl)ethyl]amine
2-(1-benzofuran-2-yl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}pyridine
4-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]benzamide
5-methyl-1-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-1,2,3,4-tetrazole
1-{3-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-fluorophenyl}ethan-1-one
[(2S,4R,5R)-5-(4-chlorophenyl)-4-[({[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}amino)methyl]-1-ethyl-2-methylpyrrolidin-2-yl]methanol
1-[2-(diethylamino)ethyl]-4-(1H-pyrazole-3-carbonyl)-1,4-diazepan-6-ol
1-cyclohexyl-4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepane
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-[2-(1H-pyrazol-4-yl)ethyl]imidazolidine-2,4-dione
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(naphthalen-2-yloxy)-N-[3-(pyridin-2-yl)propyl]propanamide
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(propan-2-yl)pyrimidine
4-(4-methyl-1H-pyrazol-1-yl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidine-4-carboxylic acid
1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-N-(pyridin-3-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
3-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indazole
1-(1H-imidazol-4-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
6-[4-(morpholine-4-sulfonyl)phenyl]quinazolin-4-amine
4-(2,6-dimethylpyridin-4-yl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}propanamide
3-{[6-hydroxy-4-(1H-imidazole-5-carbonyl)-1,4-diazepan-1-yl]methyl}benzonitrile
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
3-(2,5-difluorobenzoyl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
3-[4-(1-ethyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(2-methoxyphenyl)propanamide
1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
(cyclopentylmethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
5-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
4-methoxy-6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyrimidin-2-amine
methyl 6-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-3-(2-methylpropanamido)thieno[2,3-b]pyridine-2-carboxylate
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(3-methyl-1H-pyrazol-1-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
3-amino-1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-{1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopropan-2-yl}methanesulfonamide
5-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2-oxazole-4-carboxamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-(oxan-4-yl)-N-phenylpiperidin-3-amine
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide