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3-(azepan-1-yl)-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}propan-1-one
methyl 3-[(3,4-dimethylphenyl)methyl]-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(4-fluorophenyl)-1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidin-4-ol
1-(2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1-methylurea
1,5-dimethyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-pyrazole-4-sulfonamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]azepan-4-amine
2-[2-(dimethylamino)ethyl]-9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}thiomorpholine
(2R)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}oxolane-2-carboxamide
2-(cyclohex-1-en-1-yl)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
5-(2-chlorophenyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)furan-2-carboxamide
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-{5-[6-(dimethylamino)pyridazin-3-yl]thiophen-2-yl}ethan-1-one
6-(benzyloxy)-1-cyclohexyl-4-(3-methylfuran-2-carbonyl)-1,4-diazepan-2-one
2,6-diamino-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-ol
3-(1H-1,3-benzodiazol-1-yl)-1-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
1-[2-(dimethylamino)ethyl]-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyrrolidin-2-one
ethyl 1-ethyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(2-methoxyphenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-4-ol
3-[3-ethyl-3-(hydroxymethyl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
1-(1,4-dioxan-2-ylmethyl)-3-[2-(2-fluorophenoxy)phenyl]-1-methylurea
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-phenylpiperazine
1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 2-(1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}-N-methylformamido)acetate
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(pyrazin-2-yl)propan-1-one
(2S,4S)-4-[(diethylcarbamoyl)amino]-1-methylpyrrolidine-2-carboxamide
{3-[(3-methoxyphenyl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methanol
1-[3-(4-fluorophenyl)benzoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-cyano-N,4-dimethyl-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,6-dihydropyridine-3-carboxamide
2-{[4-(3-ethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
4-[4-(1H-pyrazol-5-yl)phenyl]pyridine
6-(5-fluoropentyl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
4-(4-chlorophenoxy)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
1-{2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-2,3-dihydro-1H-indole
6-tert-butyl-2-(2-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)methanol
2-cyclopropyl-1-{6-hydroxy-4-[(3-methylpyridin-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(2-chloro-5-fluorophenyl)-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
ethyl 4-(6,7-dimethoxy-3-{[(2-phenylethyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
methyl 2-{5-[1-(3,3,3-trifluoro-2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
N-(1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one