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4-(4-chlorophenoxy)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(2-methylpyrimidine-5-carbonyl)-8-azabicyclo[3.2.1]octane
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}({[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl})amine
3-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazol-1-yl)propanoic acid
8-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-(1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxy-2-methylpropanamide
N-[(8-methoxyquinolin-5-yl)methyl]-N,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-5-phenyl-N-(quinolin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}propan-1-one
N-[2-(2-methoxyphenyl)ethyl]-2-(4-{4-[(prop-2-en-1-yl)amino]piperidin-1-yl}phenyl)acetamide
1-(2-methoxy-6-methylphenyl)-3-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]urea
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}cyclohex-3-ene-1-carboxamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][(2,3,4-trimethoxyphenyl)methyl]amine
2-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
1'-[6-(methoxymethyl)pyrimidin-4-yl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-7-methyl-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-6-fluorophenol
(3S,4S)-4-cyclopropyl-1-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(3S,7S)-5-(5-propyl-1,3,4-thiadiazol-2-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
methyl 3-cyclopropaneamido-6-{[4-(2-methylphenyl)piperazin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1S,3R)-3-amino-N-[1-(4-chlorophenyl)cyclobutyl]cyclopentane-1-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
N,4-dimethyl-2-(piperidin-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
N-{3-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}-4-phenylbutanamide
3-cyclopropaneamido-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-4-methylbenzamide
N-methyl-2-[methyl(2-phenylethyl)amino]-N-(1-methylpyrrolidin-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(pyridin-3-yl)ethan-1-one
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(4-methoxypyrimidin-2-yl)-7-azaspiro[3.5]nonan-1-ol
3-[(3R,4S)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-methyl-6-(2-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}propyl)pyridine
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-[(4-methylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(thiophen-3-yl)-1H-imidazole
1-({[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)cyclohexan-1-ol
N'-[1-(cyclohexylmethyl)piperidin-3-yl]-N,N-dimethylbutanediamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}propanamide
6-methyl-N4-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrimidine-2,4-diamine
2-(dimethyl-1,3-thiazol-4-yl)-N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
N-[(2R,3R)-1'-(3-methylfuran-2-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-fluoropyridine
5-{[(2,4-dimethoxyphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-{[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]amino}ethyl)methanesulfonamide
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-cyclobutaneamido-N-[(3,5-dimethoxyphenyl)methyl]benzamide