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N-[2-(1H-imidazol-1-yl)ethyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-[1-(4-{cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
(2S,4S)-4-amino-1-(2-methoxyquinoline-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
N-[(3R,4S)-1-[(4-cyanophenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]methanesulfonamide
N3-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N5-[3-(propan-2-yloxy)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(dimethylamino)-N-methyl-N-(1-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-2-phenylethyl)acetamide
N,N-dimethyl-2-[4-(5-methylpyridin-3-yl)phenyl]acetamide
5,6-dimethyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine
1-[(4-chlorophenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
methyl 2-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
ethyl 3-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)heptanoate
(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-phenyl-1H-pyrazole
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[3-(pyridin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
4-[1-(5-hydroxypentyl)-1H-1,2,3-triazol-4-yl]benzoic acid
2-[(1S,5R)-6-{[(1,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
6-{[(1-hydroxycyclohexyl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1-(furan-2-ylmethyl)urea
2-hydroxy-5-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]benzamide
4-ethyl-5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
(3S,4S)-4-(1H-imidazol-2-yl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidine-3-carboxylic acid
ethyl 4-[(5-methyl-1,3,4-oxadiazol-2-yl)amino]piperidine-1-carboxylate
2-{[5-(2,5-dihydro-1H-pyrrol-1-ylmethyl)furan-2-yl]sulfanyl}pyrimidine
N-({1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(1H-indol-3-yl)propanamide
6-(2-methoxyphenyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-chloro-2-{[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)amino]methyl}quinolin-4-ol
2-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]-N-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-(4-methyl-1,4-diazepan-1-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
methyl(oxolan-3-ylmethyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-cyclopropyl-9-[(2S)-2-hydroxy-3-phenylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-1-(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-cyclohexyl-4-(pyrimidin-5-yl)benzene-1-sulfonamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
8-(1,3-dimethyl-1H-indole-2-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-(propan-2-yl)piperidine-4-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
ethyl 3-benzyl-1-(pyridine-3-sulfonyl)piperidine-3-carboxylate
2-(4-methyl-1,3-oxazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(5-fluoro-1H-indol-2-yl)methyl]methylamine
4-[(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
5-chloro-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)thiophene-2-carboxamide
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(pyrimidin-4-yl)piperidine-1-carboxamide
3-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}pyridine
2,3,5-trimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine