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3-[(2R,3R,6R)-5-[(4-fluoro-3-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
N-methyl-2-(methylamino)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[1-(thiophen-3-yl)propan-2-yl]amine
N-[2-(1-{[(5-methylpyridin-2-yl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(4-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(7-fluoro-4-methylquinolin-2-yl)ethyl]-1λ6-thiolane-1,1-dione
4-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
9-[6-hydroxy-2-(propan-2-yl)pyrimidin-4-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-({2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
N-ethyl-2,3-difluoro-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]morpholine
methyl 6-[3-(4-methylphenyl)propanoyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-1H-1,3-benzodiazole
(3aS,6aR)-5-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(2-methoxypyridin-3-yl)-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
15-methyl-N-[2-(morpholin-4-yl)ethyl]-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
6-methyl-4-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-[(3S,4R)-1-(2,3-dihydroxybenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)-N-propylpropanamide
2-[4-(2-methoxyethoxy)phenyl]pyridine-4-carboxamide
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)pyridine-4-carboxamide
3-[2-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)ethyl]phenol
(1R,7S)-N-(furan-3-ylmethyl)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-[4-ethyl-4-(hydroxymethyl)piperidin-1-yl]-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
N-(3,4-difluorophenyl)-6-[2-(methylsulfanyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,3-benzoxazole
6-ethyl-3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
N4-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(2-methoxyethyl)-4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazine
ethyl 4-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
[2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]urea
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyridin-2-amine
1-[4-(4-methylphenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
1'-[(3-methyl-1H-indol-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
N-[(2,5-difluorophenyl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
methyl 5-{[(2,3-dimethoxyphenyl)methyl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-methyl-4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
4-{[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(propan-2-yl)piperidine
1-{[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}pyrrolidin-2-one
N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
3-ethoxy-N-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
7-(1,3-benzothiazol-2-yl)-4-cyclopentyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5S,9aS,9bS)-5-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
benzyl(cyclobutylmethyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine