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2-{[3-(benzyloxy)phenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-ethyl-9-(3-fluoropyridine-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]methanol
6-({ethyl[(5-methylfuran-2-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(4,8-dimethoxynaphthalen-1-yl)methyl]-2-(ethoxymethyl)pyrrolidine
2,2-dimethylpropyl (2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
3-phenoxy-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propan-1-one
N4-[(4,6-dimethylpyrimidin-2-yl)methyl]-6-ethyl-N2,N2-dimethylpyrimidine-2,4-diamine
2-[(3-chlorophenyl)methyl]-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-diazinane-2,4-dione
2-(1H-indol-3-yl)-1-[3-(pyrrolidin-1-yl)piperidin-1-yl]ethan-1-one
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(2-methoxyethoxy)ethan-1-one
5-amino-N-[(1R,3R)-3-aminocyclopentyl]-4-phenyl-1H-pyrazole-3-carboxamide
(4aS,8aS)-2-cyclobutanecarbonyl-7-(pyridine-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
8-(3-hydroxybenzoyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-chlorophenyl)methyl]-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
2-{1-[3-(pyrrolidine-1-carbonyl)benzenesulfonyl]pyrrolidin-2-yl}-1,3-thiazole
(3S,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(thian-4-yl)butanamide
N,N-diethyl-1-(5-methyl-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
2-(3-methoxypropyl)-8-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-ethynyl-N-(3-methyl-1H-pyrazol-5-yl)benzamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1-[(2,3,4-trifluorophenyl)methyl]-1H-imidazole
methyl (1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
1-[(3S)-3-ethylmorpholin-4-yl]-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butan-1-one
4-[5-(4-methyl-1,2,3-thiadiazol-5-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(trifluoromethyl)benzamide
1-[(3-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
2-methoxy-1-{4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3-ethyl-5-[(2S)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
2-(4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-amine
2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-4-methoxyphenol
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
3-(2-acetamidopropyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-indole-2-carboxamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(trifluoromethyl)phenyl]methyl})amine
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]pyrimidin-2-amine
1-methyl-4-[(4-methyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
5-(2-cyclopentylacetamido)-N-cyclopropyl-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-amino-4-(2-chloro-4-hydroxy-5-methoxyphenyl)-6-(4-methyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
2-[2-(dimethylamino)ethyl]-9-(1H-1,2,4-triazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-oxo-1-(quinolin-3-ylmethyl)pyrrolidine-3-carboxylic acid
1-{2-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}azepan-2-one
3-(1-methyl-1H-pyrazol-5-yl)-N-[1-(thian-4-yl)piperidin-4-yl]propanamide
N-[1-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
3-{[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-1λ6-thiane-1,1-dione
1-(2-methoxy-5-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol