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N-(2-phenylethyl)-1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(phenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-indole-3-carboxamide
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(pyrimidin-4-ylmethyl)acetamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethylbenzamide
1-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]-3-methylbutan-1-ol
3-fluoro-N-[(2R,3R)-1'-(1H-indol-3-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)piperidine
N-[(3S,4R)-4-methoxyoxolan-3-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[(4-fluorophenyl)methyl]-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
7-fluoro-N-(2-hydroxy-3-phenoxypropyl)-2-methylquinoline-4-carboxamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[1-(pyrimidin-4-yl)ethyl]benzamide
3-methyl-2-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-tert-butyl-4-hydroxypyrimidine-5-carboxamide
4-(1-methyl-1H-imidazole-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R,6R)-5-(1H-indazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2R,3R)-1'-[(2,6-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
6-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)pyridine-2-carboxylic acid
2-(1H-indol-3-yl)-1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)ethan-1-one
4-(1-{2-[(thiophen-2-ylmethyl)carbamoyl]ethyl}piperidin-3-yl)benzoic acid
(3aS,6aS)-2-acetyl-5-[(2-chlorophenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]amino}propanoate
2-[4-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperazin-1-yl]-N-ethylacetamide
N-(2-methoxyethyl)-4-methyl-3-{[(2,2,2-trifluoroethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-N-(1,3-thiazol-2-yl)propanamide
5-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-phenylpiperidin-2-one
(3S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}pyrrolidin-3-ol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]pyridine-3-carboxamide
methyl 3-cyclohexaneamido-6-{[(furan-2-ylmethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-methoxy-6-[3-(methoxymethyl)-1H-1,2,4-triazol-5-yl]-N,N-bis(propan-2-yl)benzamide
1-({1-[(1-methanesulfonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)azepane
7-amino-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
2-(4-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
ethyl 4-{2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamido}piperidine-1-carboxylate
5-(2,4-difluorophenoxymethyl)-N-(3-hydroxy-3-methylbutyl)-N-methyl-1,2-oxazole-3-carboxamide
N-[2-(2-chlorophenyl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
(1-benzothiophen-2-ylmethyl)({[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
7-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-2-methyl-2,7-diazaspiro[4.5]decane
2-[4-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-ol
methyl 5-[(1-cyclohexylethyl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-(2-hydroxy-3-methylbutanoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-methoxy-6-[2-(trifluoromethyl)phenyl]pyrimidin-2-amine
7-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[(5-methylfuran-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-methoxyethyl)-1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide