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3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
2-(2-{[(1-ethyl-1H-indazol-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-8-[(4-hydroxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
N-methyl-2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(3-methoxyphenyl)amino]butanamide
(benzylsulfamoyl)(cyclopropylmethyl)(2-methoxyethyl)amine
3-(but-2-yn-1-yl)-5-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-(cyclopropylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2R,6S)-2,6-dimethyl-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}morpholine
3-methyl-5-(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[4-(furan-2-yl)phenyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxamide
1-phenyl-4-[4-(pyridin-4-yl)pyrimidin-2-yl]piperazine-2-carboxylic acid
3-methyl-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
5-cyclobutanecarbonyl-1'-(3-methylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-(thiophen-2-ylmethyl)piperidine
(1R,6S)-3-[2-(1H-imidazol-2-yl)benzoyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
1-(2-{2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
5-(diethylamino)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(2-fluorophenoxymethyl)-N-[2-(4-methylphenyl)propan-2-yl]-1H-pyrazole-3-carboxamide
2-(1H-imidazol-2-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-[(4-fluorophenyl)methyl]-5-[(2-methoxyethyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
(2S,4S)-4-amino-1-{2-[(2,3-dimethylphenyl)carbamoyl]acetyl}-N-ethylpyrrolidine-2-carboxamide
[(3R,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(3-phenylpropyl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-2-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-4-amino-N,N-diethyl-1-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
2-(2,5-dimethylphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-{1-[1-(2,4,5-trifluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[(3R,4S)-1-(2-hydroxyethyl)-4-phenylpyrrolidin-3-yl]-2-(2-oxoazepan-1-yl)acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
3-{3-cyclopentyl-5-[2-(methylsulfanyl)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(2-methoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-ol
3-(1,3-benzothiazol-2-yl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propan-1-one
{[5-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)furan-2-yl]methyl}dimethylamine
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
6-ethyl-N2,N2,N4-trimethyl-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-(1-methyl-1H-imidazol-2-yl)-1-[2-(methylsulfanyl)benzoyl]piperidine
1-methyl-5-phenyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
1-butyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-(thiophen-3-ylmethyl)urea
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,3-oxazole-5-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
1'-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one