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2-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-(4-oxo-4H-chromen-6-yl)-3-[2-(pyrrolidin-1-yl)ethyl]urea
1-methyl-8-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(hydroxymethyl)-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-ol
4-chloro-N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-[(3-methyloxetan-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-(cyclopropylsulfamoyl)-6-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-benzyl-N-(2-hydroxyethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-(3-hydroxypropyl)-1-[1-(quinolin-4-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-hydroxypropan-2-yl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[2-(4-fluorophenoxy)phenyl]-3-(hydroxymethyl)-4-methylpiperazine-1-carboxamide
(3R,4R)-N-(cyclohexylmethyl)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
1-{4-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
4-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1λ6-thiomorpholine-1,1-dione
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}propanamide
2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2-(furan-2-yl)azepane
1-cyclopentyl-4'-(2,2-dimethylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}benzoic acid
methyl (2S,4S)-1-[(2,5-dimethoxyphenyl)methyl]-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
3-(4-cyano-2-fluorophenyl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}urea
(1S,5R)-6-(cyclopropylmethyl)-3-[1-(4-methoxyphenyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-({4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
3-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
5-benzenesulfonamido-N-[(2,3-difluorophenyl)methyl]-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carboxamide
5-(3-{2-[4-(trifluoromethoxy)phenyl]-1H-imidazol-1-yl}propyl)-1H-1,2,3,4-tetrazole
2-({[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(2,2-dimethylpropyl)-3-(2-oxo-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)piperazin-2-one
N-(2-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-2-ylmethyl)-N-propylbenzamide
N,N-diethyl-3-{[(thian-4-yl)amino]methyl}pyridin-2-amine
2-[4-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenoxy]ethan-1-ol
2-{2-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenoxy}acetic acid
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methylphenol
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(pyridin-2-yl)propan-2-yl]amine
4-[4-(piperazin-1-ylmethyl)phenyl]benzamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2,6-trimethylquinoline-3-carboxamide
N-cyclopropyl-1-{1-[6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
methyl 1-{3-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
N-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}quinolin-6-yl)acetamide
2-(4-chloro-2-methylphenoxy)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-ethyl-1,2-oxazole-3-carboxamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-4-(4-methoxyphenyl)butane-1,4-dione
2-phenyl-1-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)ethan-1-ol
6-cyclopropyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine