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{1-[(3-methoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(2S)-2-amino-3-hydroxy-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
2-amino-8-[1-(propan-2-yl)piperidine-3-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(2-phenoxyethyl)-2-(pyrrolidin-1-ylmethyl)piperidine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
2-methoxy-N-[1-(2-phenylethyl)-7-(4-phenylpiperazine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
1-[(4aS,8aS)-4a-hydroxy-7-(pyrazin-2-yl)-decahydro-2,7-naphthyridin-2-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-(1H-pyrazol-1-yl)benzamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyridine-3-carbonyl)-1,4-diazepane
1-benzyl-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-6-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-9H-purin-6-amine
[(2,4-dimethoxy-3-methylphenyl)methyl](ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
4-ethyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[(3-methylpyridin-4-yl)methyl]acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2,N4-dimethyl-N2-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrimidine-2,4-diamine
N-(1-methyl-1H-pyrazol-3-yl)-2-[5-oxo-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
5-{[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
2-methyl-1-{5-[2-(morpholin-4-ylmethyl)phenyl]thiophen-2-yl}propan-1-one
(1R,5S,6R)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
(1S,5R)-6-(2-methoxyethyl)-3-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(oxane-4-carbonyl)piperidine-3-carboxylic acid
[(2,6-difluoro-3-methoxyphenyl)methyl](ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1-(3,5-dimethylphenyl)-4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperazin-2-one
methyl 3-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]benzoate
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(2,6-dimethylpyridin-3-yl)pyrimidine
1-[(4aR,8aR)-4a-hydroxy-7-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-(1-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
1-(4-{[1-(2-hydroxybutyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}thiophen-2-yl)ethan-1-one
4-(1H-pyrazol-1-yl)-6-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
3-(hydroxymethyl)-N-[3-(2-methoxyacetamido)-2-methylphenyl]morpholine-4-carboxamide
{9-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-chloro-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyridine-2-carboxamide
N-methyl-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
N5-(2H-1,3-benzodioxol-5-ylmethyl)-1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{4-[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenol
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(oxan-4-yl)piperazine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
4-{5-[(3-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
3-(2,4-dimethoxyphenyl)-1-[(4-methyl-1,4-oxazepan-6-yl)methyl]urea
6-chloro-4-(4,4-difluoropiperidine-1-carbonyl)-2-methylquinoline
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pent-4-en-1-one