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N-{1-[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
3-tert-butyl-4-(8-hydroxyquinolin-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4S)-1-(2,2-diphenylethyl)-N-methyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(2R,3R)-2-(benzyloxy)-1'-(1H-indole-6-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-[(5-acetylthiophen-3-yl)methyl]-N,N-dimethylpiperazine-1-carboxamide
(3S,4S)-4-(1H-imidazol-2-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
2-[(1S)-1-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl]-3-methylpyridine
4-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperazine-1-sulfonamide
3-(2-methylphenyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
2-[6-(8-methoxy-2-methylquinolin-5-yl)pyridin-3-yl]acetic acid
4-[2-(2-aminoethyl)quinazolin-4-yl]-3-butyl-1-methylpiperazin-2-one
[1-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
4-(4-fluorophenyl)-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-4-oxobutanamide
5-{[benzyl(methyl)amino]methyl}-N-(1,4-dioxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
5-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-methyl-3-[2-oxo-2-(3-phenylpiperidin-1-yl)ethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-(2,3,6-trimethylquinoline-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
(2S,4S)-4-(cyclooctylamino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-(3-chloropyridin-2-yl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(3S,4S)-1-[2-(2-chlorophenyl)acetyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
4-{[4-(3-chloro-1-benzothiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1-cyclopropylpyrrolidin-2-one
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-{1'-[(3-fluoro-4-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
1-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-3-[2-(ethanesulfonyl)ethyl]urea
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)pyrazolo[1,5-a]pyridine-2-carboxamide
1-(4-methylphenyl)-4-[2-(morpholin-4-yl)acetyl]piperazin-2-one
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
methyl 4-({[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl](methyl)carbamoyl}amino)-3-methylbenzoate
2-(4-acetyl-5-benzyl-2-oxopiperazin-1-yl)benzonitrile
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(naphthalen-2-ylmethyl)-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-ethyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-5-carboxamide
1,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 5-(1,3-thiazole-5-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
4-[1-(cyclopropylmethyl)-1H-pyrazol-4-yl]-1-[(4-methoxyphenyl)methyl]-1H-pyrazole
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
1-cyclopropanecarbonyl-4-[(6-methylquinolin-5-yl)methyl]-1,4-diazepan-6-ol