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N-methyl-5-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-3-carboxamide
3-{5-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-cyclohexyl-1-(2-methylpropyl)-4-oxo-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-[(tert-butylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-{3-methyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
8-(3-chlorobenzoyl)-2,8-diazaspiro[4.5]decan-3-one
9-[(4-chloro-2-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[5-(methanesulfonylmethyl)pyridin-2-yl]piperidin-4-yl}pyrrolidin-2-one
N-(2-hydroxybutyl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
4-{[1-(adamantan-1-yl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
{1-[(6-methoxy-2H-chromen-3-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
methyl 3-{[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)carbamoyl}propanoate
N-({8-[(3-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-(2-methoxy-4-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({2-[(2-chlorophenyl)methyl]morpholin-4-yl}methyl)benzoic acid
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-{3-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
N-{[7-(3-methylbut-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzenesulfonamide
methyl (2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(2,3-dimethyl-1H-indole-7-amido)pyrrolidine-2-carboxylate
4-[(3,4-difluorophenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-ethylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
4-(4-chlorophenyl)-1-{[2-hydroxy-5-(pyrazin-2-yl)phenyl]methyl}piperidin-4-ol
1-methyl-3-(2-methylpropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(2S)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-oxopiperidine-2-carboxamide
N-[(3R,4S)-1-cyclopentyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]-3-methoxypropanamide
5-(1-benzoylpiperidin-4-yl)-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-methyl-N-{1-[1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
4-benzyl-3-ethyl-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-5-one
N-[2-(4-chlorophenyl)ethyl]-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetamide
(3S,5S)-1-(2-methylfuran-3-carbonyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-3-(pyridin-3-yl)propanamide
8-fluoro-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]quinoline-2-carboxamide
ethyl 3-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-4-methylpentanoate
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-hydroxypiperidine-4-carboxylic acid
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-{[4-(2-methylpropyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[1-(pyridin-4-yl)propyl]piperidine-4-carboxamide
5-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-(2,4-dimethylpyrimidine-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)-N-(2-hydroxyethyl)propanamide
(3R,4S)-1-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
3-({4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 4-{[1-(2-methylpropyl)-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
5-(2-cyclopentylacetamido)-N,1-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide