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3-[(4-fluorophenyl)methyl]-N-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[(4-methoxypiperidin-1-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(5-methyl-1H-pyrazol-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
methyl (2R,4S)-4-hydroxy-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
N,N-dimethyl-2-[(1S,5R)-3-(6-methylpyridine-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(2-methoxyethyl)-6-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-ethyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrimidine-5-carboxamide
(4aS,7aR)-1-(3-fluorobenzenesulfonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R)-N-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)oxolan-3-amine
3-{methyl[(5-methylfuran-2-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
2-(2-cyclopropylpyrimidin-5-yl)-N-methyl-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
1-cyclopropyl-N-[3-(2,4-dimethylphenoxy)propyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-(3-chloro-4-methylphenyl)-3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
N-ethyl-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine-3-carboxamide
6-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]quinoxaline
4-(4-methyl-1H-pyrazol-1-yl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-fluoro-5-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
2-(1H-imidazol-2-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}benzamide
1-methyl-4-{[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-methylpropyl)-5-(pyridin-2-ylmethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,3,5,6-tetramethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
2,4,5-trimethyl-6-[2-(methylsulfanyl)phenyl]pyrimidine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-2-(3-phenylpiperidin-1-yl)acetamide
6-(3-chlorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[4-(propan-2-yl)phenyl]-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-[(3R,4S)-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-methoxypropanamide
N-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-2-fluorobenzamide
3-benzoyl-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(3-methylpentanoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5,8-dimethoxy-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methylquinolin-2-amine
N-[(3S,4R)-4-(propan-2-yl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]acetamide
2-(propan-2-yl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
1-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydroquinolin-2-one
8-{[3-(difluoromethoxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(oxolan-2-ylmethyl)propylamine
2-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
2-[(3,5-difluorophenyl)methyl]-8-[2-(oxolan-3-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
N,2-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]furan-3-carboxamide
3-{3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
N-(4-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
methyl 2-[(4-{4-[(2-methylpropyl)carbamoyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)sulfonyl]benzoate
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one