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2-cyclopentyl-N-{3-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-(3-methoxyphenyl)piperazin-2-one
(3R)-N-[2-chloro-5-(propylcarbamoyl)phenyl]-3-hydroxypyrrolidine-1-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2,4-triazin-3-amine
1-(cyclohexylmethyl)-3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]piperidin-2-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
1,3-dimethyl-5-({[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
4-(4-{[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}phenyl)-2-methylbutan-2-ol
N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{3-[2-(dimethylcarbamoyl)ethyl]phenyl}thiomorpholine-4-carboxamide
N-(1-{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(4-fluorophenyl)ethyl)-2-methoxy-N-methylacetamide
1-(2,2-diphenylethyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
4-cyano-1-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrrole-2-carboxamide
1-{4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-3-methoxyphenyl}ethan-1-one
N-(furan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrrole-2-carboxamide
2-methyl-2-{4-[4-(methylamino)pyrimidin-2-yl]phenyl}propanenitrile
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
[1-(2,3-dihydro-1H-inden-2-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
(1S,5R)-6-methyl-7-oxo-N-[2-(propan-2-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
8-benzyl-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]propanamide
1'-[(2S)-1-methanesulfonylpyrrolidine-2-carbonyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2R,4R)-4-hydroxy-N-{1-[(2-methylphenyl)methyl]cyclopropyl}pyrrolidine-2-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide
N-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-{4-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}methanesulfonamide
4-fluoro-N-{[1-(4-formylbenzoyl)piperidin-3-yl]methyl}benzamide
N-[(5-ethylpyridin-2-yl)methyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
N-(oxolan-2-ylmethyl)-3-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}propanamide
2-(pyridin-4-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-methyl-2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-(1-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
methyl 3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
6-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine-2-carboxamide
(4aS,7aR)-1-(3-cyclopentylpropyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(2-phenylethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(thian-4-yl)piperazine
N,N-dimethyl-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-sulfonamide
{9-benzyl-3-cyclopentanecarbonyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(3aR,6aR)-2-acetyl-5-(6-carbamoylpyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-1-(2-methylpropyl)-8-{[4-(2-methylpropyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-chloro-2-(propan-2-yloxy)phenyl]-2-(methoxymethyl)piperidine-1-carboxamide
2-[3-(5-methylfuran-2-yl)-5-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-[3-(benzyloxy)azetidine-1-carbonyl]-3-(3-methoxyphenyl)-1H-pyrazole
6-(1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
4-benzyl-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
4-hydroxy-N-[(1R,2R)-2-hydroxycyclohexyl]-2-(4-methylphenyl)-N-propylpyrimidine-5-carboxamide