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2-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
methyl (2S,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
2-(4-methylphenoxy)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
7-(1H-inden-2-yl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-1-(3-methoxypropyl)-6-{[(1s,4s)-4-aminocyclohexyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]but-2-yn-1-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyridin-3-yloxy)ethyl]pyridin-2-amine
N-[(3R,4S)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
methyl 5-[(2-ethylbutyl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-phenyl-1H-1,2,3-triazole
3-chloro-2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-indole
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-1-(2,4-difluorophenyl)-3-methyl-1H-1,2,4-triazole
6-[(3-fluorophenyl)methoxy]-4-(1-methylpiperidin-4-yl)-1-(2-methylpropyl)-1,4-diazepan-2-one
9-[2-(2-oxo-2,3-dihydro-1H-imidazol-1-yl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-({4-methyl-5-[1-(pyridazin-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N,4-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
2-(2-methoxyethyl)-9-{2-[methyl(phenyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-(piperidin-4-yl)urea
(7-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H,2H-naphtho[2,1-b]furan-2-yl)methanamine
4-(2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}ethyl)phenol
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-{2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole
N-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methanesulfonamide
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-methoxy-N-(pyridin-4-ylmethyl)benzamide
(4aR,7aS)-1-propyl-4-(quinoline-8-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-chlorophenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(prop-2-en-1-ylsulfanyl)acetamide
2-(4-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}piperazin-1-yl)acetic acid
5-methyl-N-[(2-methylphenyl)methyl]-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5,6-dimethyl-2-(4-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-methyl-7-(4-methylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3R,5S)-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-benzyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
1-(3-hydroxyazetidin-1-yl)-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
2-(4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(furan-2-ylmethyl)piperazin-2-yl)ethan-1-ol
2-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(3-hydroxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-cyclohexyl-2-(6-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propan-1-ol
2-{[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(4-methylphenyl)pyrimidin-2-yl](methyl)amino}ethan-1-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2S,4S)-4-(2,3-dihydro-1,4-benzodioxine-6-amido)-N-ethyl-1-propylpyrrolidine-2-carboxamide
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one