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2-methoxy-6-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
5,6-dimethyl-2-oxo-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
5-hydroxy-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]pyrazine-2-carboxamide
(1R,5R)-6-(1-benzofuran-2-ylmethyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-2-yl)propan-1-ol
(3S)-4-(5-chloropyridine-3-carbonyl)-3-ethylmorpholine
2-{[(5-methoxyfuran-2-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-cyclopentanecarbonyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxamide
(3S,4S)-1-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-(1H-indol-7-ylmethyl)-1λ6-thiane-1,1-dione
(2S,4S)-4-amino-N,N-diethyl-1-[2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidine-2-carboxamide
3-[(2R,3R,6R)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(2-amino-1,3-thiazol-4-yl)-1-(4,4-difluoropiperidin-1-yl)propan-1-one
N-{[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidin-3-yl]methyl}-2,2-dimethylpropanamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]piperidin-3-yl]methanol
1-{3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-[1-methyl-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}({[1-(morpholin-4-yl)cyclopentyl]methyl})amine
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
4-[5-(hydroxymethyl)furan-2-carbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1,5-dimethyl-4-[(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-ethyl-3-{[2-(furan-2-ylmethyl)-3-hydroxypropyl]sulfamoyl}-N-methylbenzamide
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclohex-3-ene-1-carboxamide
methyl 3-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}benzoate
1-(1-benzylpiperidin-4-yl)-N-(1,3-dihydroxypropan-2-yl)piperidine-3-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)urea
1-{9-[(1-ethyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.6]dodecan-3-yl}-2-methoxyethan-1-one
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
(2E)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methylpent-2-enamide
N,1-dimethyl-2-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]imidazolidine-4-carboxamide
3-butyl-4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-methylpiperazin-2-one
6-chloro-2-{[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
1,3-dimethyl-N-[2-(1,3-thiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-{4-[2-(pyrrolidin-1-yl)ethyl]phenyl}urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
methyl 3-propanamido-5-({[2-(1H-pyrazol-1-yl)phenyl]formamido}methyl)benzoate
6-(2-{[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]amino}ethyl)pyrimidin-4-ol
3-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-6-methylpyridazine
N-(3-acetylphenyl)-4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazine-1-carboxamide
4-hydroxy-N-(oxolan-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-methyl-1,2-oxazole-4-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(methylsulfanyl)acetamide
3-[(3R,4S)-1-(2-methyl-2-phenylpropanoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[1-(thian-4-yl)piperidin-4-yl]quinoxaline-6-carboxamide
{1-[(3-ethoxy-4-methoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1-methylpiperidin-4-ol
2-amino-N-[(3-chlorophenyl)methyl]-3-ethyl-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide