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8-methoxy-N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-chloro-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]propanamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
2-(2-hydroxyphenoxy)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
2-{2-methyl-3-[({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
4-(azepan-1-yl)-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(4aS,7aR)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]cyclohexane-1-carboxamide
2-(2-{[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]amino}ethyl)-3,4-dihydroquinazolin-4-one
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(2,3-dimethoxyphenyl)methyl]propanamide
1-[(3,4-dimethylphenyl)methyl]-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
(4aR,7aS)-1-[(5-ethylpyridin-2-yl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-hydroxyethyl)-3-{5-[2-(methylsulfanyl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-ethyl-1-(1H-imidazol-1-ylmethyl)-N-[1-(4-methoxyphenyl)propyl]cyclopropane-1-carboxamide
[(2S,4R)-1-methyl-4-{[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}pyrrolidin-2-yl]methanol
1-cycloheptyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(8-chloroquinolin-2-yl)methyl](methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(5-fluoropyridine-3-carbonyl)piperidine-4-carboxylic acid
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-(furan-2-ylmethyl)-2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
9-{[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-5-ethyl-2,6-dimethylpyrimidine
(4S)-4-hydroxy-3,3,4-trimethyl-N-(2-phenylethyl)piperidine-1-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-chloropyridine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(thiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(quinolin-6-ylmethyl)acetamide
N-[4-({[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-{1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
5-methyl-N-({1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N-[2-(benzyloxy)ethyl]-1-cyclopentylpiperidine-3-carboxamide
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenol
4-[4-(2-fluoro-4-methoxyphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-(1H-1,2,3-benzotriazol-5-yl)-4-(1-hydroxy-3-phenylpropyl)piperidine-1-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3,4-dimethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidin-3-yl}methyl)benzamide
methyl 3-acetamido-5-({[5-(hydroxymethyl)furan-2-yl]methyl}amino)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
N,1-diethyl-3-methyl-N-[2-(2-methylphenoxy)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(5-methyl-1H-pyrazol-1-yl)propanamide
3-cyclopropyl-1-(2,3-dimethylphenyl)-5-[2-(1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
1-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethyl)azepan-2-one
methyl[3-(methylsulfanyl)propyl]{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-benzyl-8-(oxan-4-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({3-methyl-7-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)ethane-1-sulfonamide
N-[(3R,4S)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide