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9-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-1-[1-methyl-4-(oxolan-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]ethan-1-one
methyl (2S,4R)-4-(dimethylamino)-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]pyrrolidine-2-carboxylate
2-(3-fluoro-4-methoxyphenyl)-2-[(1H-imidazol-2-ylmethyl)(methyl)amino]acetic acid
(1S,5R)-6-(2-methoxyethyl)-3-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
1-propyl-3-(pyrrolidine-1-carbonyl)-5-[4-(thiophene-2-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole
2-[({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amino]propan-1-ol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(naphthalene-2-carbonyl)pyrrolidin-3-yl]methanol
5-tert-butyl-3-{[4-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-[(2-methylphenyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[ethyl({[(3S,4R)-4-(hydroxymethyl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-[(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazol-5-yl)methyl]-1H-1,3-benzodiazole
N-(2,3-dichlorophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
4-{4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-chloro-3-(4-phenyl-1H-imidazol-5-yl)phenol
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-{4-[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
1-methyl-4-[4-(thiophen-2-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(3-{[(cyclopropylmethyl)(2-methoxyethyl)carbamoyl]amino}phenyl)-N-methylacetamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(2,5-dimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
6-methyl-3-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-4H-chromen-4-one
5-cyclopropanecarbonyl-1'-(4-fluoro-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(5-methylfuran-2-yl)ethyl]propanamide
N-{[7-(adamantane-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-amino-4-ethyl-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-1,3-thiazole-5-carboxamide
(1S,5R)-3-(4-methoxybenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(2-methyl-4-phenylpyridin-3-yl)formamido]acetamide
6-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-1H-indole
(1R,5S,8R)-3-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-tert-butyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
5-cyclopropyl-N-(3-ethoxypropyl)-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
1-{4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
6-methyl-2-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
2-(3-methyl-3-phenylpiperidine-1-carbonyl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
(4aS,7aR)-4-[(5-methylfuran-2-yl)methyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-yl]-2-hydroxyacetamide
N-[2-(4-methoxyphenyl)ethyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
(1-{[4-(4-fluorophenyl)phenyl]methyl}piperidin-2-yl)methanol
6-oxo-1-(2-phenylethyl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
5-(2,6-dimethoxyphenyl)-3-[3-(methoxymethyl)piperidin-1-yl]-1,2,4-triazine
4-[(2-fluorophenyl)methyl]-3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one