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9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{[4-(2-methylpropyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{[(4-methylphenyl)(pyridin-4-yl)methyl]amino}propane-1,3-diol
1-[(3-chlorophenyl)methyl]-4-(2-methoxypyridine-4-carbonyl)piperazine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
6-(1-benzothiophen-3-yl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-(2-fluorophenyl)-5-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{[3-(difluoromethoxy)phenyl]methyl}piperidine
8-[2-(1H-pyrazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-N-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
1-(1,3-benzoxazol-2-ylmethyl)-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
ethyl 5-{[(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazol-7-yl)formamido]methyl}furan-2-carboxylate
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-[(1-ethyl-1H-indol-3-yl)sulfanyl]ethan-1-one
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(methanesulfonylmethyl)piperidine
3-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]benzoic acid
(2S,4R)-4-amino-1-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
5-[(3,3-diphenylpiperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
1-butyl-3-(2-hydroxypyridin-3-yl)-1-(pyridin-3-ylmethyl)urea
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(cyclopropylmethyl)piperazine
2,4-dimethyl-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}-1,3-thiazole-5-carboxamide
7-[5-(oxolan-2-yl)thiophene-2-carbonyl]-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-{4-[(3-{[1-(3-fluorobenzoyl)piperidin-4-yl]oxy}-4-methoxyphenyl)methyl]piperazin-1-yl}ethan-1-one
8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-5-(morpholin-4-ylmethyl)-N-[1-(1,3-thiazol-5-yl)ethyl]furan-3-carboxamide
3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}-1-(furan-3-carbonyl)piperidine
4-{4-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-fluorophenyl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
3-{[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-6-methyl-1,2-dihydropyridin-2-one
1-cyclohexyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-4-carboxamide
11-{[(3,5-difluorophenyl)methyl]amino}-4-[3-(propan-2-yloxy)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 1-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
3-ethyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{[(9H-fluoren-9-yl)amino]methyl}-4-(pyridin-3-yl)phenol
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-methylphenoxymethyl)piperidine
(cyclohex-1-en-1-ylmethyl)[1-(1H-imidazol-1-yl)propan-2-yl]amine
(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
N-[2-(methylsulfanyl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,6-dimethylpyridine-4-carboxamide
N-[(2-methoxyphenyl)methyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-(4-phenoxybenzoyl)piperidine-1-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(1-methylcyclopropyl)propanoyl]piperidine-2-carboxamide
N-(5-chloro-2-methylphenyl)-N'-methyl-N'-[2-(morpholin-4-yl)propyl]propanediamide
4,4-difluoro-1-({2-[3-(piperidin-1-yl)propoxy]phenyl}methyl)piperidine
N-cyclohexyl-N,5-dimethyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N,N-dimethyl-5-{[(2-methylphenyl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}cyclohexanecarboxamide
dimethyl({4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine