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5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(3-methylbutan-2-yl)pyridin-2-amine
2-(1H-1,3-benzodiazol-1-yl)-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]propanamide
3-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrrole
1-(1-benzylpiperidin-4-yl)-4-ethyl-1,4-diazepan-5-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-(3-methylphenoxy)-1-[1-(piperidin-4-yl)pyrrolidine-2-carbonyl]piperidine
1-(4-ethylpiperazin-1-yl)-3-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propan-1-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2,2-bis(hydroxymethyl)butan-1-one
2-amino-6-(2-hydroxypropan-2-yl)-4-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}pyridine-3-carbonitrile
8-[(4-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-6-methylquinolin-4-ol
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,4-dimethyl-1,3-thiazole
(3aR,7aS)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-8-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2,4,5-trifluoro-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-(adamantan-1-yl)-2-[2-(azepan-1-ylmethyl)-4-(pyrimidin-2-yl)phenoxy]acetamide
1-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-{[(3-chloro-5-fluoro-4-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}butan-1-ol
1-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
N-(9H-fluoren-9-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,4-diazepan-6-ol
4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydroquinazolin-2-one
(2E)-1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
N-methyl-3-(2-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-1-{2-[(3-methylpyridin-4-yl)amino]ethyl}urea
4-cyclopropyl-6-[4-(pyridin-3-yl)piperazin-1-yl]pyrimidine
2-ethyl-4-phenyl-9-(pyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecane
methyl[3-(oxolan-2-yl)propyl]{[2-(trifluoromethoxy)phenyl]methyl}amine
N-(2,2-diphenylethyl)-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N-methyl-2-(3-phenyl-1H-1,2,4-triazol-5-yl)-N-(thiophen-3-ylmethyl)acetamide
6-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
6-methoxy-4-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-(2-{[(1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-{2-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(3-hydroxy-3-methylbutyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)benzamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
3-{2-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
methyl 6-(2-phenylpropyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(2-hydroxyethyl)(methyl)sulfamoyl]-N-methylbenzamide
(2S,4S)-4-amino-1-(5-fluoro-2-methoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
2-methoxy-5-{1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidine