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N-cyclopropyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
3-({7-[(1-propyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propan-1-one
{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N-(2,3-dihydro-1-benzofuran-3-yl)-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-(4-chloro-1-ethyl-1H-pyrazol-5-yl)-1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazole
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(4-phenyloxan-4-yl)methyl]acetamide
N-(4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(1H-pyrazol-1-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-{2-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-1-methylimidazolidine-2,4-dione
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
7-(2-hydroxyethyl)-2-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
(7S,9aR)-N-benzyl-7-[(2S)-butan-2-yl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-cyclopentyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide
1-(cyclobutylmethyl)-4-(furan-2-carbonyl)-1,4-diazepane-6-carboxylic acid
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
2-(3-oxopiperazin-1-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
N-tert-butyl-5-chloro-2-({1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
3-{[(2,2-difluoroethyl)amino]methyl}-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-methoxyacetamide
3-(3-hydroxy-3-methylbutyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-fluoroquinazolin-4-amine
3-[(2-methyl-1H-indol-5-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
2-benzyl-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1,3-thiazole-4-carboxamide
3-methyl-8-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-1,2,4-triazol-1-yl)acetamide
1-cyclopentyl-4-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
(3S)-3-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}azepan-2-one
(2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)urea
3-(5-methylfuran-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-[(4-{[3-(propan-2-yl)-1,2,4-thiadiazol-5-yl]carbamoyl}phenyl)methyl]piperidine-3-carboxamide
N-cyclopropyl-2-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-4-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(3-phenylpropyl)amine
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
ethyl 1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-2-carboxylate
4-benzyl-1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-ethyl-1,4-diazepan-5-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
1-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{[3-(trifluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aS)-5-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(1H-imidazol-2-yl)ethyl]acetamide
5-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid