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2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
N,3-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
2-benzyl-8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
3-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-phenylurea
3-({[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}methyl)-N,N-dimethylpyridin-2-amine
2-methyl-N-[3-(6-methyl-9H-purin-9-yl)phenyl]propanamide
1-[3-(1-methylpiperidin-3-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
2-methyl-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl}-1-methyl-1H-1,3-benzodiazole
1-cyclohexanecarbonyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrrolidine-2-carboxamide
N-({8-[(3,4-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-{[3-methyl-7-(thiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}oxolane-2-carboxamide
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1λ6-thiomorpholine-1,1-dione
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
N-(4-{4-[(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
2-{4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-{2-[4-(2,4-difluorophenyl)piperazin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-{[3-(cyclopentyloxy)phenyl]methyl}-2,5-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-methyl-N-[2-(2-methyl-1H-indol-3-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-methoxyethyl)-1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-(1H-imidazol-2-yl)-1-[4-(2-methoxyphenyl)phenyl]-1H-imidazole
(3S,4R)-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(3,4-difluorophenyl)methyl]-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
2-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
{1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-cycloheptyl-4-{4-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(2-methoxyphenyl)ethyl]amine
4-[(2,5-dimethoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2,2-dimethylcyclopropanecarbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
N-[2-(2-phenoxyethoxy)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
1-(5-cyclopropyl-1H-pyrazole-3-carbonyl)-4-methanesulfonyl-1,4-diazepane
5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methoxybenzamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3,3-diphenyl-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
8-[(3-hydroxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,N-dimethyl-3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methanesulfonamidoacetamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-(3,3,3-trifluoropropyl)-2,8-diazaspiro[4.5]decane
4-(3,6-dimethylpyrazin-2-yl)-2-[(3-methoxyphenyl)methyl]morpholine