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2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}quinoxaline
3-(3-cyano-4-methylphenyl)-1-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)urea
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-4-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)butanamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazole
5-(hydroxymethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]furan-2-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-(4-chlorophenyl)-N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}-5-methylphenol
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(pyridine-2-carbonyl)piperazine
3-[(3R,4S)-1-[(3-chloro-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(4aS,7aR)-1-[(4-chlorophenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,4-diazepan-5-one
5-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-3-methyl-1H-pyrazole-4-carboxamide
(2S,3R)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxybutanamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(dimethylamino)-N-[3-(3-methoxyphenyl)phenyl]azepane-1-carboxamide
4-hydroxy-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
(1S,6R)-9-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,5S)-5-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1-methylpyrrolidin-3-amine
8-(1-aminocyclopropanecarbonyl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-fluoro-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
(3S,4S)-1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-4-methylpiperidine-3,4-diol
3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-{2-[(5-ethylpyrimidin-2-yl)(methyl)amino]ethyl}cyclopentan-1-ol
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(4aS,8aR)-1-butyl-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl](oxolan-3-ylmethyl)amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3,5-dichlorophenyl)methyl]pyrrolidin-3-yl]methanol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-({1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3,4-tetrazol-5-yl}(phenyl)methyl)morpholine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]thiophene-3-carboxamide
2,6,6-trimethyl-1-(2-methylpropyl)-3-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
3-(1-methylpiperidin-2-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propan-1-one
3-[2-(piperidin-2-yl)ethyl]-5-(quinoxalin-2-yl)phenol
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
1-methyl-5-{3-methyl-1-[(3-methylphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-imidazole
{2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}urea
3-ethyl-4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-[(2-phenylphenyl)carbamoyl]piperidin-3-yl]propanoic acid
5-[4-(2,1,3-benzoxadiazol-5-ylmethyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N3-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methylpyridine