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2-[1-(2-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-cyclopropylpyrimidine
N-(butan-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{[2-(2-methoxyphenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-ol
6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-1H-pyrrolo[2,3-b]pyridine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamide
methyl 3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)benzoate
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
6-(4-chlorophenyl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(4-{[3-(propan-2-yloxy)propyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(4-chlorophenyl)methyl]-N-[(3-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
[1-({1-[5-(3-methylphenyl)furan-2-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(4aS,8aR)-6-[2-(benzyloxy)acetyl]-1-butyl-decahydro-1,6-naphthyridin-2-one
1-[3-(5-chloro-2-methoxyphenyl)propyl]-1H-imidazole
(R)-cyclohexyl[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methanol
1-cyclopentyl-3-(3-methoxyphenyl)-3-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-6-(piperidine-1-carbonyl)pyrazine
1-{[4-(cyclopentyloxy)phenyl]methyl}-4-[(dimethylamino)methyl]azepan-4-ol
4-[(2-methyl-6-propylpyrimidin-4-yl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
2-(3-methyl-1,2-oxazol-5-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
N-{[1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
3-hexyl-8-(5-methylpyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
(3S)-4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(1-propylpiperidin-4-yl)piperidine
3-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}pyridin-2-amine
N-cyclopropyl-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazine-2-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
ethyl 2-({[(1R,5S,6R)-3-(furan-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}(methyl)amino)acetate
1-(6-methoxyquinolin-8-yl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
N-(3-methoxypropyl)-2-methyl-N-(1-methylpiperidin-4-yl)-5-(propan-2-yl)furan-3-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
(3aR,6aS)-1-oxo-5-(3-phenyl-1,2-oxazole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
dimethyl(2-{2-[1-(quinoline-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-[2-(dimethylamino)-1-phenylethyl]-1-(2-hydroxyethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
4-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-4-oxobutane-1-sulfonamide
(4aS,8aS)-2-(2,3-dihydro-1-benzofuran-5-ylmethyl)-decahydroisoquinolin-4a-ol
2-methyl-4-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)butan-2-ol
1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[(2R,3R)-1'-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
9-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-3-oxa-9-azaspiro[5.5]undecane
2-chloro-4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
4-{3-[2-(2-chloro-4-fluorophenyl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1H-pyrazole
2-(5-{[(2S)-2-benzyl-3-oxopiperazin-1-yl]methyl}furan-2-yl)benzonitrile
1-methyl-3-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
N-cyclohexyl-1-(cyclohexylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide