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(3R,4R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-cyclopropyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)benzamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-(4-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrazine
diethyl({4-[(3S)-3-ethylmorpholine-4-carbonyl]-5-phenylfuran-2-yl}methyl)amine
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-(morpholin-2-ylmethyl)urea
{4-benzyl-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}methanol
N-cyclopropyl-N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
2-(ethylsulfanyl)-5-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]pyrimidine
3-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
5-(2-chlorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]furan-2-carboxamide
1-(2-aminoacetyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
ethyl 4-[2-(2-phenylethyl)morpholin-4-yl]piperidine-1-carboxylate
N-{1-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}acetamide
2-({[2-(3-fluorophenyl)ethyl]amino}methyl)-4-(pyridin-2-yl)phenol
5-(quinolin-8-yl)pyrimidin-2-amine
3-cyclopropyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
(3-{[(2-methanesulfonylethyl)amino]methyl}-2,4,6-trimethylphenyl)methyl acetate
N-[2-(1H-indol-3-yl)ethyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
4,6-dimethyl-2-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(5-propyl-4H-1,2,4-triazol-3-yl)urea
(2S,4S)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[(4-phenylphenyl)methyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
methyl 3-methyl-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3,5-dimethyl-2-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1H-indole
N-(dicyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1λ6-thiomorpholine-1,1-dione
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-4,6-dimethyl-2H-pyran-2-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(6-methylpyridin-2-yl)piperazine
2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-2-one
9-[2-(2,4-dimethylphenoxy)ethyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-[(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]acetamide
N-[5-(dimethylamino)pentyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(cyclopropylmethyl)-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-{8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-(3-methoxyphenyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
4-phenyl-1-(prop-2-yn-1-yl)-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
2-methoxy-1-[1'-(2-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
5-benzenesulfonamido-1-ethyl-2-methyl-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
4-(cyclohexylmethyl)-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
2-(4-{[4-(cyclopentyloxy)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol