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(3S,4R)-1-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
ethyl 1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
1-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)-4-methylpiperazine
6-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
2-(4-{3-[(4-fluorophenyl)methoxy]phenyl}-1H-pyrazol-1-yl)-N-methylacetamide
2-[4-(2,2-diphenylethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
(3S,9aR)-8-(2,5-difluorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-chloro-2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}quinoline
5-ethenyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(4-methoxyphenyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-phenylpropanamide
N-[(2R,3R)-1'-cyclopentanecarbonyl-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-ethyl-1-(3-methanesulfonamido-4-methoxyphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]urea
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)butan-2-ol
2-cyclohexyl-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-amino-4-[3-(methylsulfanyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
1-(2-methoxyethyl)-6-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
(1-benzothiophen-2-ylmethyl)[(4-{[1-(2-fluorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]methylamine
N-ethyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
8-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(2-methyl-1,3-thiazol-4-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[cyclopentyl(methyl)amino]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)acetamide
N,3,6,7-tetramethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[3-(4-methyl-1,3-thiazol-5-yl)propyl]amine
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
[3-(3-methylbut-2-en-1-yl)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]methanol
1-[6-hydroxy-4-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
2-amino-6-cyclopentyl-4-[4-(2-hydroxyethoxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-tert-butyl-N-[(3R,4S)-1-(2-hydroxyethyl)-4-propylpyrrolidin-3-yl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide
4-{7-[(2-fluorophenyl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholine
1-[1-(3-fluorobenzenesulfonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-tert-butyl-5-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-{5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(2-methylquinolin-4-yl)-7-azaspiro[3.5]nonan-1-ol
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(3,4,5-trimethoxyphenyl)acetamide
4-{2-[(2-methoxyethyl)carbamoyl]ethyl}-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
3-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3,9-diazaspiro[5.6]dodecan-10-one
1-tert-butyl-4-{[methyl(4-methylquinazolin-2-yl)amino]methyl}pyrrolidin-2-one
4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-methylbutan-1-one
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2-methoxyphenyl)methyl]piperidine
N5-(1-benzylpyrrolidin-3-yl)-1-cyclopentyl-N3,N3-diethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(1-benzyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)pyridine
5-methyl-1-(4-methylphenyl)-4-[3-(piperidin-1-yl)propanoyl]piperazin-2-one