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N-(oxolan-2-ylmethyl)-2-[4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-2-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
2-fluoro-5-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}benzamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
2-(3-methyl-4-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-(carbamoylmethyl)-N-[3-(2-fluorophenyl)propyl]piperidine-3-carboxamide
(3R,9aR)-8-[(2,4-dimethylphenyl)methyl]-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-(1-ethyl-1H-pyrazol-4-yl)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
2-{3-[2-amino-3-cyano-6-(5-methylfuran-2-yl)pyridin-4-yl]phenoxy}acetamide
1-(7-fluoro-2-methylquinoline-4-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
4-[(4-chlorophenyl)methyl]-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-phenylprop-2-en-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-amino-1-[(3-methyl-1,2-benzoxazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
N,N-dimethyl-2-[(1S,5R)-6-[(2-methylnaphthalen-1-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-[4-(1-methyl-1H-imidazol-2-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-8-fluoroquinoline
2-(4-methoxy-3-methylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
4-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
2-[2-(azepan-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-3-(4-methoxyphenyl)-1H-pyrazole
2-(4-methyl-1H-imidazol-5-yl)-1-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-imidazole
1-cycloheptyl-N-methyl-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}-4-(2-phenylethyl)piperazin-2-one
3-(azocan-1-yl)-N-[(1-methyl-1H-pyrazol-5-yl)methyl]propanamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-3,5-difluorobenzamide
5-{1-[(5-chlorothiophen-2-yl)methyl]pyrrolidin-2-yl}-N-(2-methoxyethyl)thiophene-2-carboxamide
N-(4-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-imidazol-2-yl}phenyl)acetamide
1-{2-oxo-2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyridin-2-one
N-[2-(4-hydroxyphenyl)ethyl]-2-[(3-methoxyphenyl)amino]butanamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(4aR,7aS)-1-methyl-4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-methylpiperazine-1-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
4-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-N-methyl-1,3-thiazol-2-amine
1-methoxy-8-[1-(3-methoxyphenyl)propan-2-yl]-1,8-diazaspiro[4.5]decan-2-one
1-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-(pyridin-3-yloxy)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
3-(3-cyano-1H-pyrazol-4-yl)benzoic acid
2-{4-chloro-2-[1-(thiophen-3-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
methyl 3-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamido]azepane-1-carboxylate
2-(4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one