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(1R,9S)-5-amino-3-(4-chlorophenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]acetamide
(1H-imidazol-2-ylmethyl)(methyl){[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
(3S,4S)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-{methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}pyrrolidin-3-ol
6-(3-chlorophenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4S)-4-amino-1-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3,5-dimethyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
(1-{1-[6-(2-methoxyphenyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyridin-2-yl]piperidin-4-yl}piperidin-3-yl)methanol
3-(2-methoxyphenyl)-N-[2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
4-(1H-indole-6-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
6-(3-chlorophenyl)-2-(2-methylpyrrolidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}propanamide
8-[(3-fluoro-2-methylphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2,1,3-benzothiadiazol-4-yl)-4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carboxamide
3-(5-methylfuran-2-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
methyl(naphthalen-1-ylmethyl)[(3-{2-[4-(pyridine-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
[(1-benzylpiperidin-4-yl)methyl]({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
5-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3,4-dihydropyrimidin-4-one
3-(2-methylpropyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
1-(2-cyclohexylethyl)-3-hydroxy-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
ethyl 2-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)acetate
3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
1-{[2-(benzyloxy)phenyl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[(3-fluorophenyl)methyl]-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
6-{3-oxo-3-[2-(2-phenylethyl)morpholin-4-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N'-(2-ethoxyphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]propanediamide
8-(cyclohexylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(furan-3-ylmethyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazin-2-yl]ethan-1-ol
3-[3-(1-ethyl-1H-pyrazol-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-amino-1-(2-benzyl-1,3-thiazole-4-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[2-(morpholin-4-ylmethyl)phenyl]urea
N-(isoquinolin-5-ylmethyl)-N,5-dimethyl-1,2-oxazole-3-carboxamide
3-[(diethylamino)methyl]-N-(1-ethyl-1H-pyrazol-5-yl)benzamide
2-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)benzonitrile
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
2-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N-[2-(diethylamino)ethyl]-4-{[(2-fluorophenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidin-2-one
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
6,7-dimethyl-4-[({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]-2H-chromen-2-one
5-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-methoxyethyl)propanamide
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-cyclohexyl-N-[2-(methylsulfamoyl)ethyl]-1H-pyrazole-4-carboxamide
2-(3-hydroxypropyl)-9-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one