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6-[2-(3-methoxyphenoxy)ethyl]-1,2-dihydroisoquinolin-1-one
3-(4-benzylpiperidine-1-carbonyl)-1-cyclopentyl-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
3-[(4-fluorophenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-methyl-5-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrimidin-2-amine
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-ethoxyethan-1-one
1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-4-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,4-diazepan-2-one
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3-ethoxypropyl)propanamide
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carboxamide
2-{2-methoxy-5-[(4-sulfamoylpiperazin-1-yl)methyl]phenoxy}acetic acid
N-(2-{[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
2-methyl-5-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]pyrimidin-4-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-(1-hydroxyhexan-2-yl)-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-phenoxyethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,3-thiazol-2-amine
5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-thiazole-5-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
9-(5-chloro-3-fluoropyridin-2-yl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methoxyphenyl)-1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]propan-1-one
N-(1-{1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
1-(4-{[4-(3,5-difluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
1-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
(1R,5R)-6-(cyclopropylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-ethyl-4-(4-methylpiperazin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-methylbut-2-en-1-one
N-[2-(furan-2-yl)ethyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl}-4-methylpyrimidine
2-{4-[(3,5-difluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
3-(2-chlorophenyl)-N-cyclopropyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
3-(5-{[(butan-2-yl)(cyclopentyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
(5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-1,3-benzodiazol-2-yl)methanol
N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
1-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
ethyl 2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)(methyl)amino]acetate
1-cyclopentyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-[(3-chlorophenyl)methyl]-3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide