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N-ethyl-1-methyl-N-(oxan-4-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
5-(2-methoxyacetamido)-1-methyl-N-[3-(methylsulfanyl)propyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
7-[(2,6-difluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(1-{1-[(2,5-dimethylthiophen-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N,2-dimethyl-7-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
ethyl 4-{6-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-(1-{1-[2-(naphthalen-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
8-(2-hydroxyethyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]benzoic acid
2-[methyl(pyridin-3-ylmethyl)amino]-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
3-chloro-5-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1,2-dihydropyridin-2-one
4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-1H-pyrrole-2-carbonitrile
1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
2,6-difluoro-3-methoxy-N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]benzamide
3-[(4aR,8aR)-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-{2-[1-(2,4-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
3-methyl-1-[2-(2-methylpropoxy)phenyl]-3-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}urea
5-(2-chloro-4-methoxyphenoxymethyl)-N-ethyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
6-{[methyl(oxan-4-yl)amino]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
5-(2,6-difluorophenoxymethyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(4-ethanesulfonamidobenzoyl)piperazine-2-carboxylic acid
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
8-methyl-2-propyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(3-chlorophenyl)-4-(2-hydroxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(1H-imidazol-1-yl)propyl]-2,7,8-trimethylquinoline-4-carboxamide
N,5-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-({[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amino}methyl)pyrrolidin-3-ol
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
[3-(hydroxymethyl)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methanol
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-[2-(1H-indol-3-yl)ethyl]-6-(1-phenyl-1H-pyrazole-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
4-methyl-7-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)-2H-chromen-2-one
[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)methylamine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
5-{[benzyl(methyl)amino]methyl}-N-[2-(1H-imidazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
7-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-5-methoxy-1H-indazole
N-cyclobutyl-2-{4-[2-(2,4-difluorophenyl)acetyl]morpholin-3-yl}acetamide
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-methoxyphenyl)piperidine
N-[1-(3-methylphenyl)piperidin-4-yl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
4-[(dimethylamino)methyl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azepan-4-ol