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N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
5-ethyl-6-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-3-methyl-1,2,4-oxadiazole
5-methyl-N-[(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentanecarbonyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-oxobutanamide
3-(4-methyl-1H-pyrazol-1-yl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-(2-fluorophenyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2,2-dimethylcyclopropane-1-carboxamide
2-[1-(3-methylpyridin-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrazine
2-[3-benzyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(carbamoylmethyl)acetamide
1-(2,6-difluorobenzoyl)-3-(4-methoxyphenoxymethyl)piperidine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
1'-(2,3-dihydro-1-benzothiophene-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(4-oxo-4-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}butan-2-yl)acetamide
1-[(3-methylphenyl)methyl]-5-[1-(pyrrolidin-1-yl)propan-2-yl]-1H-1,2,4-triazole
6-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-chloro-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-{4-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-4-oxobutyl}acetamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
N-[2-(methylsulfanyl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-(5-methylfuran-2-yl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
(1S,4S)-5-(3-chlorobenzoyl)-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 3-acetamido-1-ethyl-5-{[1-(2-methoxyphenyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}acetamide
5-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-1H-imidazole-4-carboxylic acid
8-[(2S)-2-amino-4-hydroxybutanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1H-pyrazol-4-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-cyclopentyl-3-methyl-4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-chlorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
8-(1,3-benzothiazol-2-yl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-1,8-diazaspiro[4.5]decane
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
2-{2-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(2-methylpropyl)-4-[4-(naphthalen-1-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-[2-methyl-4-(4-methylphenyl)-5-oxopiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-N,4-dimethyl-1,3-thiazol-2-amine
(2-{2-[1-(2-methoxy-4-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[(2R)-1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-oxobutan-2-yl]acetamide
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
4-(1-ethyl-1H-imidazol-2-yl)-N-[2-(propan-2-yl)phenyl]piperidine-1-carboxamide
3-(2-methoxyphenoxy)-1-[2-(trifluoromethyl)benzoyl]azetidine
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione