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2-(2,5-dimethylphenoxy)-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(propan-2-yl)pyrimidine-5-carboxamide
5-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-amine
4-(5-methylpyridin-2-yl)-1-[4-(piperidin-3-ylmethyl)benzoyl]piperidin-4-ol
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]sulfamoyl})amine
(4aR,7aS)-1-(2-methylpropanoyl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[2-(dimethylamino)ethyl]-6-(2,5-dimethylfuran-3-yl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(dimethylamino)-N-{[1-(dimethylamino)cycloheptyl]methyl}-2-(4-fluorophenyl)acetamide
1-(2-aminoethyl)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
2-[5-(3-chloro-4-methylphenyl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl]acetamide
2-ethyl-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
4-(2-methoxypyridin-3-yl)-3-methylpyridine
8-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[5-(2-methoxy-5-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
6-hydroxy-N-[3-(3-phenylpropoxy)phenyl]-1,4-oxazepane-4-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-(2-ethyl-1H-1,3-benzodiazol-6-yl)urea
2-(4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazin-1-yl)phenol
5-methoxy-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-4-oxo-1,4-dihydropyridine-2-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-(3-hydroxypropyl)-9-[4-(2-methylpropyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(2-methoxyphenyl)benzoyl]-2-(trifluoromethyl)morpholine
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
(1S,4R)-2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2-azabicyclo[2.2.1]heptan-3-one
3-(2,4-dimethoxybenzoyl)-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidine
5-[2-(methylsulfanyl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(cyclohex-1-en-1-ylmethyl)-2-{4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]morpholin-3-yl}acetamide
4-(2H-1,3-benzodioxol-4-ylmethyl)-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenol
2-methyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1-(5-methanesulfonamido-2-methylphenyl)-3-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-5-(5-methylfuran-2-yl)-1,2,4-triazine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[1-(1-cycloheptylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(naphthalen-1-yl)ethan-1-one
N-(3-phenylprop-2-yn-1-yl)-N-propylpyrrolidine-3-carboxamide
3-{1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidin-4-yl}phenol
1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-ethoxy-5-(2-{[2-(1H-pyrazol-1-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
1-(2,4-difluorophenyl)-5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-1H-1,2,4-triazole
4-(2-methyl-1H-imidazol-1-yl)-1-[(2E)-3-phenylprop-2-enoyl]piperidine-4-carboxylic acid
N,1-dimethyl-3-(propan-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
2-amino-6-(2,2-dimethylcyclopropyl)-4-[5-(hydroxymethyl)furan-2-yl]-5-methylpyridine-3-carbonitrile
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one