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(3S,7S)-5-(5-methylthiophene-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(cyclopropylmethyl)-N-propyl-3-(quinolin-8-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,3-dihydro-1H-isoindole
2-amino-N-(1,3-dihydroxypropan-2-yl)-4-phenylpyrimidine-5-carboxamide
9-methoxy-3-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
methyl 2-(2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamido)acetate
N2-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-methylpyrimidine-2,4-diamine
methyl 4-(5-methyl-4-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-1,3-oxazol-2-yl)benzoate
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepane
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
4-ethyl-3-{[1-(2,4,6-trimethylbenzoyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(4-methoxyphenyl)propyl]-6-[(propan-2-yl)amino]pyridine-3-carboxamide
6-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-1,4-oxazepan-6-ol
2,5-dimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1,3-thiazole-4-carboxamide
1-({methyl[1-(pyridin-4-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N5-[2-(3-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,6S)-4-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}-2,6-dimethylmorpholine
N-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
N-(3-hydroxypropyl)-4-methyl-3-oxo-N-(pyridin-4-ylmethyl)-3,4-dihydroquinoxaline-2-carboxamide
1-(2-methylbenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-methyl-6-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
ethyl 5-(1H-indole-6-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(4-methyl-1H-imidazol-2-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2-[1-(2,2,6,6-tetramethylpiperidin-4-yl)piperidine-3-carbonyl]pyridine
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
7-fluoro-N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-3-methyl-1H-indole-2-carboxamide
1-(2-methoxybenzenesulfonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
methyl 2-(3-methylbutyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
6-(1,2-diphenylethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]methyl}piperidin-3-ol
2-methoxy-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
3-{1-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-1H-imidazol-2-yl}phenol
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(3,4-dimethylphenyl)ethan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-azaspiro[2.5]octane-1-carboxamide
1-(2,2-dimethyloxane-4-carbonyl)-4-(1H-imidazol-2-yl)piperidine
N'-(2-methylphenyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanediamide
methyl (2S,4R)-4-[3-(4-fluorophenyl)benzamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxylate
N-[(dimethyl-1,3-oxazol-4-yl)methyl]-3-(4-fluorophenyl)-3-phenylpropanamide
1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(methoxymethyl)piperidine
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[1-(adamantan-1-yl)piperidin-3-yl]-N-cyclopropylpropanamide
2-(2-methoxyethyl)-9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-({[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
7-[(2,3-difluorophenyl)methyl]-2-(pentan-3-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(1H-imidazol-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
methyl 1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carboxylate