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N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[5-(dimethyl-1,2-oxazol-4-yl)-1H-indol-1-yl]acetamide
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-(quinoxalin-2-ylmethyl)acetamide
N-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methanesulfonamide
4-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
N-(3-{[(butan-2-yl)(pyridin-2-ylmethyl)carbamoyl]amino}-4-methylphenyl)-2-methoxyacetamide
N-[(1-{[5-(2-cyanophenyl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
1-cyclopentyl-5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
(2R,6R)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,8-naphthyridine-2-carboxamide
dimethyl[1-(5-methylfuran-2-yl)-2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl]amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(1H-pyrazol-1-yl)benzamide
2-(methylsulfanyl)-5-({4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyrimidine
8-[2-(pyridin-4-ylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(6-methylquinolin-5-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
(3S,7S)-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-ethyl-4-({[1-(methoxymethyl)cyclopropyl](methyl)carbamoyl}amino)-N-phenylbenzamide
4-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
4-{2-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}morpholine
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-1,3-benzothiazole
3-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
8-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-4-methylpyridine
2-{[4-(1-methyl-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}oxane-4-carboxamide
1-methyl-3-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[(2-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(4-{[(1S)-1-phenylpropyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}azepane-2-carboxamide
N-[(4-methoxyphenyl)methyl]-1,5-bis(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4R)-N,N-dimethyl-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-propylpyrrolidin-3-amine
N,1,3-trimethyl-N-{1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-5-carboxamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1,5-dimethyl-4-{[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-pyrrole-2-carbonitrile
6-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
2-(2-aminopyrimidin-5-yl)-N-ethyl-6,8-dimethyl-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
3-butanamido-N-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}benzamide
N-(oxan-3-yl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-(2-methanesulfonamidoethyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-cyclohexyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
6-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-ethyl-3-{4-phenyl-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-5-yl}piperidine