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4-hydroxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(azocan-1-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
6-[9-acetyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyrazine-2-carboxylic acid
3-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
(3S,4S)-3-({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
(3R,4R)-1-(4-methoxybenzoyl)-4-{[(3-methylpyridin-2-yl)methyl]amino}pyrrolidin-3-ol
1-({3-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidin-4-ol
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(thiophen-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)propanamide
3-{2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[(2R,4S,6R)-2-(3-hydroxyphenyl)-6-(2-methylpropyl)oxan-4-yl]acetamide
N-benzyl-N-methyl-3-{1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidin-4-yl}propanamide
N-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
1-[4-(1H-imidazol-1-yl)phenyl]-N-[3-(methylamino)propyl]piperidin-4-amine
1-methyl-4-{5-[5-(oxolan-2-yl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-ol
9-methoxy-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-hydroxypropyl)-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluoro-4-hydroxyphenyl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
2-[4-(4-phenylphenyl)-1H-pyrazol-1-yl]ethan-1-ol
N'-[(3,4-dimethoxyphenyl)methyl]-N,N-dimethyl-N'-(pyridin-2-ylmethyl)butanediamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)acetamide
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-[(3S,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-({[3-(dimethylamino)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
1-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-3-(dimethyl-1,2-oxazol-4-yl)urea
(3aS,6aS)-5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
3-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]piperidine-1-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-butyl-N-methylacetamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
3-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-3-phenylpropanamide
(2E)-N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)-3-(thiophen-2-yl)prop-2-enamide
5-acetyl-N-cyclopropyl-2,4-dimethyl-N-(3-phenylprop-2-yn-1-yl)-1H-pyrrole-3-carboxamide
3-methyl-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3-[3-(oxolan-2-yl)propyl]urea
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-N-(1,3-thiazol-2-yl)thiophene-2-carboxamide
methyl 3-cyclobutaneamido-5-[(3-methylbutyl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(pyridin-4-ylmethyl)-8-(quinoxalin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrazine
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{[4-(dimethylamino)oxan-4-yl]methyl}urea
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-1,2-oxazole-3-carboxamide