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2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]ethan-1-one
(4aS,7aR)-1-(2-propoxyacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(hydroxymethyl)-9-[(4-methoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
2-methyl-7-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N5-[2-(3-chlorophenyl)ethyl]-N3-(cyclopropylmethyl)-1-(2-methoxyethyl)-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
8-methoxy-3-(pyridin-4-ylmethyl)-3,4-dihydroquinazolin-4-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(3-methoxyphenyl)methyl]amine
3-{1-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-4-(2-methoxyethyl)-4H-1,2,4-triazole
N-[2-(2-chlorophenyl)ethyl]-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}methanesulfonamide
4-chloro-2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-2-yl)methyl]amine
5-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-phenyl-1H-pyrazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1H-indol-1-yl)ethyl]benzamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pent-4-enamide
1-benzyl-3-methyl-5-(2-methylbutyl)-1H-1,2,4-triazole
4-({2-[1-(2-methyloxolane-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
6-ethoxy-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinolin-2-ol
N3-(1-methoxybutan-2-yl)-1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,7aR)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
7-fluoro-N,3-dimethyl-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1-[4-({4-[(2,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
(1S,5R)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-cycloheptanecarbonyl-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
{4-[(2-chlorophenyl)methyl]-1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}methanol
N-[2-(4-methoxyphenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-chloropyridin-3-yl)-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]urea
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(2-methoxyphenyl)propanamide
1-methyl-1'-[2-(oxan-2-ylmethoxy)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
6,7-difluoro-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-[(1S,5R)-6-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-ethyl-5-{[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,3,4-thiadiazole
1-butyl-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-methylpropanamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
3-phenyl-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-(oxolan-2-ylmethyl)-9-(1-phenylcyclopropanecarbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[(3R,4R)-4-(hydroxymethyl)-1-[(6-methoxynaphthalen-2-yl)methyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-benzyl-9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-cyclopentyl-N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-methyl-2-(2-phenyl-1H-imidazol-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide