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N-benzyl-N-(2-hydroxyethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-hydroxy-3-({[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
6-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(quinoline-6-carbonyl)piperidine-3-carboxylate
5-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3,4,7-trimethyl-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1H-indole
8-[(2R)-2-hydroxypropanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-[({[(4-fluorophenyl)methyl]carbamoyl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[4-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)piperazin-1-yl]propanamide
5-{5-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{4-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}acetic acid
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methylpyrazine-2-carboxamide
9-(1,4-dioxan-2-ylmethyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2H-indazol-2-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5-methylthiophene-2-carboxamide
(1R,5R)-3-methanesulfonyl-6-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(4-fluorophenyl)acetamide
3-methyl-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}but-2-en-1-one
2-{1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}pyridine
(2S,4R)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(methylsulfanyl)acetamido]-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 3-benzyl-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-3-carboxylate
5-methyl-N-[1-(thiophen-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(1-ethoxyethyl)phenyl]-N,6-dimethylpyrimidin-4-amine
1-(4-methyl-1H-imidazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpiperidine-4-carbonyl)piperidine
1-(3-chlorophenyl)-4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-cyclopropyl-3-(3-fluorophenyl)-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}benzamide
4-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
5-(3-methoxyphenoxymethyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-3-carboxamide
7-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-methoxyphenyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-N'-cyclopentylbutanediamide
4-fluoro-N-({1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}methyl)benzamide
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
4-[4-(2-chlorobenzoyl)piperazin-1-yl]-2-[(2,3-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-(quinoline-6-carbonyl)-1,4-oxazepan-6-ol
2-[1-(3-methylbut-2-en-1-yl)-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-methoxyethoxy)ethan-1-one
N-cyclopropyl-4-methoxy-2-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
2-(2-methoxyphenoxy)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(hydroxymethyl)azepan-4-ol
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-propoxyethan-1-one
5-fluoro-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-1H-indole-2-carboxamide
methyl 2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-[(5-fluoro-2-methylphenyl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide