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2-[(2,3-dihydro-1-benzofuran-5-ylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-ethyl-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-(4-methoxy-2-methylphenyl)-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
3-(2,3-dihydro-1H-inden-2-yl)-8-(2,2-dimethylpropyl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-[5-methyl-6-(3-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperazine
2-{3-cyclopentyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-ethyl-4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}pyrrolidin-2-one
2-methoxyethyl 2-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxylate
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-phenoxyethyl)acetamide
2-(3-methoxypropyl)-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-benzyl-2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
4-[4-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperazin-1-yl]-6-methylpyrimidin-2-amine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-benzyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,3-benzoxazole
N-(1-{4-[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-decahydro-2,7-naphthyridine-2-sulfonamide
2-[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-2-yl]ethan-1-ol
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxymethyl)furan-2-carboxylic acid
6-[4-(furan-2-yl)benzoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
7-(1-methylpiperidine-3-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
1-(3-{[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)-6-methyl-1,2-dihydropyridin-2-one
N-ethyl-6-methoxy-3-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(4-fluorophenyl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-cyclooctyl-2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)acetamide
5-[(3-methoxyphenyl)methyl]-5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-3-methylimidazolidine-2,4-dione
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(9aS)-N-(4-cyanonaphthalen-1-yl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(methylsulfanyl)ethyl]acetamide
(2R,6R)-10-methoxy-4-(1-methylpiperidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-(6-methylpyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-{3-[4-(dimethylamino)phenyl]propanoyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-1,4-diazepane
N-({7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-1-methylpiperidine-3-carboxamide
1-(2,3-dihydro-1H-indol-1-yl)-2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
4-chloro-2-[(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
[1-({1-[(1-methyl-1H-pyrrol-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
1-(2-{[1-(cyclohexylmethyl)piperidin-3-yl]amino}pyrimidin-4-yl)piperidin-4-ol
2-fluoro-N-[2-(furan-2-yl)ethyl]-6-methoxybenzamide
2-[4-(1-acetylpiperidine-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile