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8-(2-fluoro-6-methoxyphenyl)quinolin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2,3,6-trimethylquinoline-4-carboxamide
4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-3-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}pyridine
methyl N-{[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamoyl]methyl}carbamate
4-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
1-({5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-2-ol
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(pyridin-3-yl)morpholine
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2,4-dimethylpyrimidine
2-methyl-8-[(5-methylnaphthalen-1-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine
5-{3-[(2,6-dichlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}piperidin-2-one
6-methoxy-2-oxo-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(4-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyrazine
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-2-(1,3-thiazol-4-yl)acetamide
2-(cyclohexylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholine
N-(4-{[1-(2-methoxyethyl)-3-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
1-[(4aR,8aS)-1-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-[(4-methoxyphenyl)methyl]-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
3-(furan-2-yl)-3-phenyl-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
4-(dimethyl-1,2-oxazol-4-yl)-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2E)-3-(2-chlorophenyl)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)prop-2-enamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
5-benzyl-5-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
7-(furan-3-ylmethyl)-2-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-methoxy-N,3-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
4-(1H-1,3-benzodiazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3-methoxy-4-methylphenyl)formamido]acetic acid
N-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-fluoro-3-methylbenzene-1-sulfonamide
2-(4-fluorophenyl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
1-(3-chlorophenyl)-4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperazine
2-methyl-4-{4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]piperidin-1-yl}-5-propylpyrimidine
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
N,N-dimethyl-1-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)pyrrolidin-3-amine
2-phenyl-6-(2,4,5-trimethylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-(ethoxymethyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-[2-(4-ethoxyphenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(propan-2-yl)-2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propanamide
(4aS,7aR)-1-(3-fluorobenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(2,4-difluorophenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 5-(cyclohexylamino)-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
N-[1-(1-benzoylpiperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-({5-[1-(2-hydroxyethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[4-(3-methoxypropyl)piperazin-1-yl]propan-1-one
6-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile