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N-[1-(4-chlorophenyl)cyclobutyl]oxane-2-carboxamide
3-[(4-fluorophenyl)methyl]-N-[furan-2-yl(phenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-3-yl)benzamide
1-[2-(dimethylamino)ethyl]-6-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
5-cyclopropyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1,3,4-oxadiazol-2-amine
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(1-phenylcyclopropyl)acetamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1-benzofuran-2-carboxamide
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
2-(2,4-diethoxy-3-methylphenyl)-1H-imidazole
(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
4-{2-[2-(trifluoromethyl)phenyl]ethyl}-4H-1,2,4-triazole
4-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3R,9aR)-8-(4-methylbenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(2H-1,3-benzodioxole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3R,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-phenylpyrrolidin-3-amine
1-methoxy-8-(quinolin-4-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}oxane-4-carbonitrile
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
4-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)-N-[(2-fluorophenyl)methyl]benzamide
4-(5-methylpyridin-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-4-ol
N-(2-{4-[(3,3-dimethylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)oxolane-2-carboxamide
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}morpholin-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
(4aR,7aS)-1-benzyl-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,5-dimethoxybenzamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
3-methyl-N-{1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
9-(3-hydroxypyridine-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(3-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]-N-methylbenzamide
5-(3,4-dimethylphenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-(1,2-oxazol-3-ylmethyl)propanamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{2-[3-(1H-pyrazol-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
2-{5-methyl-4-[(5-methylfuran-2-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(4-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propanamide
1-(3-chlorophenyl)-4-(5-fluoro-2-methoxybenzoyl)-5-methylpiperazin-2-one
N-cyclopropyl-6-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(1R,2R)-1-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1H-inden-2-yl]acetamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(2-phenoxyacetyl)piperidine-3-carboxylate
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide