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(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(3-methoxypropanoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
3-(3-methoxy-4-methylphenyl)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propan-1-one
3-{4-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
ethyl 5-[(5-acetamidothiophen-2-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 4-(4-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-1-yl)benzoate
2,6-dihydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
4-(2,2-diphenylethyl)-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
(5S,9aS,9bS)-5-(4-hydroxy-3-methoxyphenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
3-(2-chlorophenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
3-(5-methylfuran-2-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
3-(3-fluoro-4-methoxybenzoyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
3-{1-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]piperidin-4-yl}benzonitrile
[(3-{[1-(2-fluorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-cyclohexyl-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-(2-ethylpiperidine-1-carbonyl)-N-(3-hydroxy-2,2-dimethylpropyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-methoxy-6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridazine
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzothiazole-6-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-methoxy-N-(2-methoxyethyl)acetamide
7-[(4-fluorophenyl)methyl]-2-{[5-(methoxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decane
1-acetyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]piperidine-4-carboxamide
3-[1-(2-methoxyacetyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
{2-[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
1-(3-fluorophenyl)-4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
1-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(1R,5R)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
(5S,9aS,9bS)-5-(3-hydroxyphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2R,3S)-3-hydroxy-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]butanoic acid
3-(azepane-1-carbonyl)-N-[(5-chlorothiophen-2-yl)methyl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2,3,6-trifluorobenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-{4-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-methyl-N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
[1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-4-phenylpiperazine
N-cyclopropyl-N-(2-phenyl-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
1-cyclopropanecarbonyl-4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepan-6-ol
3-fluoro-N-{[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
(4aR,7aS)-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
(3aR,6aS)-5-[5-(methoxymethyl)furan-2-carbonyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
N-cyclopropyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)cyclohexanecarboxamide
4-({1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-2-yl}methyl)morpholine
2,6-dimethyl-5-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(5-chlorothiophen-2-yl)methyl]-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide