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1-[2-(2-methoxy-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)ethyl]pyrrolidine
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]quinoxaline
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-(3-methyl-1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
3-(2-methylpropyl)-2-oxo-1-[2-(pyrrolidin-1-yl)propyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(3aR,6aR)-2-cyclopentyl-5-[3-(1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-ethyl-5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}urea
8-(3-fluoro-2-methoxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-(3-phenoxypropanoyl)piperazin-2-one
N-(furan-2-ylmethyl)-3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(methylsulfanyl)-N-(oxolan-2-ylmethyl)acetamide
2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(furan-2-ylmethyl)acetamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyrazine-2-carboxamide
5-{1-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-[4-(methylsulfanyl)benzoyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}urea
3-(1H-pyrazol-1-ylmethyl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]benzamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
(2R,3R)-1'-[3-(1H-pyrazol-1-yl)propyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(oxan-3-yl)sulfamoyl]-N-(thiophen-2-ylmethyl)benzamide
(1H-imidazol-2-ylmethyl)({[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl})methylamine
ethyl 1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[3-(thiophen-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-[2-(2,3-dimethylphenoxy)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
N-ethyl-2-[4-(quinolin-3-yl)phenyl]acetamide
4-[3-(1-methyl-1H-pyrazol-4-yl)propanamido]-N-phenylpiperidine-1-carboxamide
N-(4-ethoxy-2-fluorophenyl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
3-(2-fluorophenyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
(3S,9aR)-3-methyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-methyl-10-oxo-N-(quinolin-6-yl)-3,9-diazaspiro[5.6]dodecane-3-carboxamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
2-(ethylsulfanyl)-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]-N-methylbenzene-1-sulfonamide
5-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]pyrrolidin-2-yl}thiophene-2-carboxylic acid
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyridin-2-yl)piperazine
methyl[(2,3,4-trimethoxyphenyl)methyl][(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
2-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}-5-methylpyrazine
2-(3-methyl-1,2-oxazol-5-yl)-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-{3-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one