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2-[(3-methyl-1H-pyrazol-4-yl)formamido]-N-(2-methylphenyl)acetamide
1-methyl-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine-2-carboxylic acid
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
ethyl (1R,5S,6R)-3-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate
2-[3-methyl-5-(1-oxo-1,2-dihydroisoquinolin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]quinoline-3-carboxamide
8-fluoro-2-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)methyl]quinolin-4-ol
2-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-({7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
7-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-2,7-dioxo-1,3-diazepane-4-carboxamide
4-methyl-2-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]-1,2-dihydrophthalazin-1-one
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(1,3-thiazol-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
dimethyl[1-(3-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}phenyl)ethyl]amine
3-(2,1,3-benzothiadiazol-5-ylmethyl)-3,4-dihydropteridin-4-one
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methyl-3-(methylsulfanyl)propanamide
7-(2-fluoro-6-methoxyphenyl)-1,2-dihydroisoquinolin-1-one
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
2-[5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-(propan-2-yl)-1H-1,3-benzodiazole
N-methyl-1-(piperidin-3-ylmethyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidine-2-carboxamide
5-{5-[(methylsulfanyl)methyl]furan-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine-3-carboxylate
1-[(1-{6-[methyl(propan-2-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(4-methoxyphenyl)-3-methyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyridin-3-yl)ethan-1-one
{[3-(2-{4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethylpropanamide
3-(oxolan-2-ylmethyl)-5-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(4-methoxyphenyl)-3-methyl-4-phenylmethanesulfonylpiperazin-2-one
3,5-dimethoxy-N-({1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
1-{5-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]thiophen-2-yl}ethan-1-one
N-[(3-chlorophenyl)methyl]-3-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]propanamide
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-[2-oxo-2-(3-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
1'-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
1,9-dimethyl-4-(morpholine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
N2-benzyl-6-(2,3-difluorophenyl)-1,3,5-triazine-2,4-diamine
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N-[2-(2-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(2E)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(4-methoxyphenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]prop-2-enamide
5-(2-cyclopentylacetamido)-N,1-dimethyl-N-[(4-methylphenyl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
[4-benzyl-1-(quinolin-8-ylmethyl)piperidin-4-yl]methanol
6-{2-[4-phenyl-5-(quinolin-8-yl)-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
4-benzyl-3-ethyl-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,4-diazepan-5-one