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N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
[(3,4-dimethoxyphenyl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
5-methoxy-2-[(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
[(3R,4R)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carboxamide
(4aS,7aR)-1-[(4-phenoxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyrimidine
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
N-(1-methyl-1H-pyrazol-4-yl)-2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}acetamide
3-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(furan-2-ylmethyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-5-[2-(oxolan-2-yl)ethyl]-1H-1,2,4-triazole
3-methyl-4-(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
N-[3-(1H-indazol-1-yl)propyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-{[1-(1-acetylpiperidine-3-carbonyl)azetidin-3-yl]oxy}benzoic acid
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-methyl-1,3-benzoxazole-6-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-4-oxo-4H-chromene-2-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
2-methoxy-5-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
(4aS,7aR)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1-phenylpiperazin-2-one
2-{3-[(4-methoxyphenyl)methyl]-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
(2-{3-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]phenoxy}ethyl)dimethylamine
methyl 3-(3,5-dimethylbenzoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(dimethylamino)butanamide
(3aR,6aR)-2-(oxane-4-carbonyl)-5-(pyridin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-(4-methylpiperidine-1-carbonyl)piperidine
9-[2-(3-chloro-4-fluorophenoxy)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
{6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-yl}methanamine
6-oxo-N-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
thiophen-2-yl(1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidin-4-yl)methanol
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[(2-chlorophenyl)methyl]-4-(3-methylfuran-2-carbonyl)morpholine
N-({1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}methyl)cyclopropanecarboxamide
2-methyl-N-(1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
2-amino-4-(2-methylphenyl)-6-(pyridine-4-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(3-fluorophenyl)-4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)piperazin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-(3-chloro-4-hydroxyphenyl)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one