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3-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-ol
(3aR,6aR)-2-(2-methoxyethyl)-5-(pentylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2,1,3-benzoxadiazol-4-ylmethyl)[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]ethylamine
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-[3-(dimethylamino)propyl]-N-methyl-1-[2-(methylsulfanyl)benzoyl]piperidin-3-amine
[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-(9-methyl-9H-carbazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-ethyl-N,4-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-1,3-oxazole-5-carboxamide
5-chloro-N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-methyl-N-{2-[(1-methylpiperidin-4-yl)amino]ethyl}methanesulfonamide
3-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1-methyl-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-benzyl-1-cyclopropyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-[5-(2,3-dihydro-1H-inden-1-ylmethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
6-[(1-benzyl-1H-imidazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
1-benzyl-4-[2-(4-methylphenoxy)acetyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
methyl 4-(5-methyl-4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
3-cyclopentyl-1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]propan-1-one
N-cyclopropyl-2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
N-({7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-cyclooctyl-2-[(2-hydroxyethyl)(1,3-thiazol-2-ylmethyl)amino]acetamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
2-(2-aminoacetyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-hydroxy-2-(pyridin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidine-5-carboxamide
[3-(2-phenylethyl)-1-(quinolin-8-ylmethyl)piperidin-3-yl]methanol
1-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-[1-(5-chloro-2-methoxybenzoyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
5-{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-(3,4-dihydro-2H-1,4-benzoxazine-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
6-({[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)-2-methylpyrimidin-4-ol
(2S,4S)-4-amino-N-(propan-2-yl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
N-[2-(2-ethyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
N-benzyl-N,1-dimethyl-5-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1R,5S,6S)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-3-azabicyclo[3.1.0]hexane
2-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propan-2-ol
2-(dimethylamino)-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-2-(4-methylphenyl)acetamide
4-[2-(2-methylphenyl)benzoyl]-2-(trifluoromethyl)morpholine
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-cyano-2-ethylphenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
[3-(4-fluorophenoxy)propyl](methyl)[(2-methyl-2H-indazol-3-yl)methyl]amine
[(2R)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl]methanol
5-{1-[2-(dimethylamino)benzoyl]pyrrolidin-2-yl}-N,N-dimethylthiophene-2-carboxamide